Tsuyoshi Adachi - Search Results

Year	Number of Results
2002	1
2004	1
2006	2
2008	1
2012	1
2015	1
2016	1
2017	1
2018	2
2019	2
2020	2
2021	5
2022	2
2023	5
2024	4

1

Soft ground micro TBM jack speed and torque prediction using machine learning models through operator data and micro TBM-log data synchronization.

Kilic K, Narihiro O, Ikeda H, Adachi T, Kawamura Y. Kilic K, et al. Among authors: adachi t. Sci Rep. 2024 Apr 27;14(1):9728. doi: 10.1038/s41598-024-60681-8. Sci Rep. 2024. PMID: 38678078

2

Optimization Efforts for Identification of Novel Highly Potent Keap1-Nrf2 Protein-Protein Interaction Inhibitors.

Otake K, Hara Y, Ubukata M, Inoue M, Nagahashi N, Motoda D, Ogawa N, Hantani Y, Hantani R, Adachi T, Nomura A, Yamaguchi K, Maekawa M, Mamada H, Motomura T, Sato M, Harada K. Otake K, et al. Among authors: adachi t. J Med Chem. 2024 Mar 14;67(5):3741-3763. doi: 10.1021/acs.jmedchem.3c02171. Epub 2024 Feb 26. J Med Chem. 2024. PMID: 38408347

3

Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development.

Maeba T, Hirata K, Kotoku M, Seki N, Maeda K, Hirashima S, Yamanaka H, Sakai T, Obika S, Hori A, Hara Y, Noji S, Suwa Y, Yokota M, Fujioka S, Yamaguchi T, Katsuda Y, Hata T, Miyagawa N, Arita K, Nomura Y, Taniguchi T, Asahina K, Aratsu Y, Naka Y, Adachi T, Nomura A, Akai S, Oshida SI, Pai S, Crowe P, Bradley E, Steensma R, Tao H, Fenn M, Babine R, Li X, Thacher S, Soeta T, Ukaji Y, Shiozaki M. Maeba T, et al. Among authors: adachi t. J Med Chem. 2024 Jan 25;67(2):952-970. doi: 10.1021/acs.jmedchem.3c01933. Epub 2024 Jan 3. J Med Chem. 2024. PMID: 38170624

4

Discovery of Novel NLRP3 Inflammasome Inhibitors Composed of an Oxazole Scaffold Bearing an Acylsulfamide.

Ohba Y, Adachi K, Furukawa T, Nishimaru T, Sakurai K, Masuo R, Inami T, Orita T, Akai S, Adachi T, Usui K, Hamada Y, Mori M, Kurimoto T, Wakashima T, Akiyama Y, Miyazaki S, Noji S. Ohba Y, et al. Among authors: adachi t. ACS Med Chem Lett. 2023 Nov 10;14(12):1833-1838. doi: 10.1021/acsmedchemlett.3c00433. eCollection 2023 Dec 14. ACS Med Chem Lett. 2023. PMID: 38116417

5

Screening approaches for the identification of Nrf2-Keap1 protein-protein interaction inhibitors targeting hot spot residues.

Asano W, Hantani R, Uhara T, Debaene F, Nomura A, Yamaguchi K, Adachi T, Otake K, Harada K, Hantani Y. Asano W, et al. Among authors: adachi t. SLAS Discov. 2024 Mar;29(2):100125. doi: 10.1016/j.slasd.2023.11.001. Epub 2023 Nov 5. SLAS Discov. 2024. PMID: 37935317 Free article.

6

Fragment-Based Discovery of Novel VE-PTP Inhibitors Using Orthogonal Biophysical Techniques.

Asano W, Yamanaka K, Ohara Y, Uhara T, Doi S, Orita T, Iwanaga T, Adachi T, Fujioka S, Akaki T, Ikegashira K, Hantani Y. Asano W, et al. Among authors: adachi t. Biochemistry. 2023 Jul 18;62(14):2161-2169. doi: 10.1021/acs.biochem.3c00079. Epub 2023 Jul 6. Biochemistry. 2023. PMID: 37414577

7

Methyl and Fluorine Effects in Novel Orally Bioavailable Keap1-Nrf2 PPI Inhibitor.

Otake K, Ubukata M, Nagahashi N, Ogawa N, Hantani Y, Hantani R, Adachi T, Nomura A, Yamaguchi K, Maekawa M, Mamada H, Motomura T, Sato M, Harada K. Otake K, et al. Among authors: adachi t. ACS Med Chem Lett. 2023 Apr 7;14(5):658-665. doi: 10.1021/acsmedchemlett.3c00067. eCollection 2023 May 11. ACS Med Chem Lett. 2023. PMID: 37197451

8

The discovery of 3,3-dimethyl-1,2,3,4-tetrahydroquinoxaline-1-carboxamides as AMPD2 inhibitors with a novel mechanism of action.

Kitao Y, Saito T, Watanabe S, Ohe Y, Takahashi K, Akaki T, Adachi T, Doi S, Yamanaka K, Murai Y, Oba M, Suzuki T. Kitao Y, et al. Among authors: adachi t. Bioorg Med Chem Lett. 2023 Jan 15;80:129110. doi: 10.1016/j.bmcl.2022.129110. Epub 2022 Dec 20. Bioorg Med Chem Lett. 2023. PMID: 36563792

9

Structure-based drug design of novel and highly potent pyruvate dehydrogenase kinase inhibitors.

Bessho Y, Akaki T, Hara Y, Yamakawa M, Obika S, Mori G, Ubukata M, Yasue K, Nakane Y, Terasako Y, Orita T, Doi S, Iwanaga T, Fujishima A, Adachi T, Ueno H, Motomura T. Bessho Y, et al. Among authors: adachi t. Bioorg Med Chem. 2021 Dec 15;52:116514. doi: 10.1016/j.bmc.2021.116514. Epub 2021 Nov 10. Bioorg Med Chem. 2021. PMID: 34808405

10

Exploring the optimal reverse supply chain for e-waste treatment under Chinese government subsidy.

Wang J, Li W, Mishima N, Adachi T. Wang J, et al. Among authors: adachi t. Waste Manag. 2022 Jan 1;137:128-138. doi: 10.1016/j.wasman.2021.10.031. Epub 2021 Nov 6. Waste Manag. 2022. PMID: 34752946

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