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Correction to "An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline".
Aprile S, Colombo G, Serafini M, Di Paola R, Pisati F, Bhela IP, Cuzzocrea S, Grosa G, Pirali T. Aprile S, et al. Among authors: pirali t. ACS Med Chem Lett. 2023 Nov 27;14(12):1891-1892. doi: 10.1021/acsmedchemlett.3c00497. eCollection 2023 Dec 14. ACS Med Chem Lett. 2023. PMID: 38116440 Free PMC article.
Deuterium in drug discovery: progress, opportunities and challenges.
Di Martino RMC, Maxwell BD, Pirali T. Di Martino RMC, et al. Among authors: pirali t. Nat Rev Drug Discov. 2023 Jul;22(7):562-584. doi: 10.1038/s41573-023-00703-8. Epub 2023 Jun 5. Nat Rev Drug Discov. 2023. PMID: 37277503 Free PMC article. Review.
First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy.
Angeli A, Micheli L, Carta F, Ferraroni M, Pirali T, Fernandez Carvajal A, Ferrer Montiel A, Di Cesare Mannelli L, Ghelardini C, Supuran CT. Angeli A, et al. Among authors: pirali t. J Med Chem. 2023 Jan 26;66(2):1616-1633. doi: 10.1021/acs.jmedchem.2c01911. Epub 2023 Jan 10. J Med Chem. 2023. PMID: 36626645 Free PMC article.
An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline.
Aprile S, Colombo G, Serafini M, Di Paola R, Pisati F, Bhela IP, Cuzzocrea S, Grosa G, Pirali T. Aprile S, et al. Among authors: pirali t. ACS Med Chem Lett. 2022 Jul 14;13(8):1278-1285. doi: 10.1021/acsmedchemlett.2c00166. eCollection 2022 Aug 11. ACS Med Chem Lett. 2022. PMID: 35978700 Free PMC article.
CIC-39Na reverses the thrombocytopenia that characterizes tubular aggregate myopathy.
Cordero-Sanchez C, Pessolano E, Riva B, Vismara M, Trivigno SMG, Clemente N, Aprile S, Ruffinatti FA, Portararo P, Filigheddu N, Zaggia I, Bhela IP, Serafini M, Pirali T, Colombo MP, Torti M, Sangaletti S, Bertoni A, Genazzani AA. Cordero-Sanchez C, et al. Among authors: pirali t. Blood Adv. 2022 Aug 9;6(15):4471-4484. doi: 10.1182/bloodadvances.2021006378. Blood Adv. 2022. PMID: 35696753 Free PMC article.
STIM1 and ORAI1 mutations leading to tubular aggregate myopathies are sensitive to the Store-operated Ca2+-entry modulators CIC-37 and CIC-39.
Riva B, Pessolano E, Quaglia E, Cordero-Sanchez C, Bhela IP, Topf A, Serafini M, Cox D, Harris E, Garibaldi M, Barresi R, Pirali T, Genazzani AA. Riva B, et al. Among authors: pirali t. Cell Calcium. 2022 Jul;105:102605. doi: 10.1016/j.ceca.2022.102605. Epub 2022 May 18. Cell Calcium. 2022. PMID: 35636153 Free article.
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