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Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer's disease.
Eur J Med Chem. 2021 Jan 15;210:113059. doi: 10.1016/j.ejmech.2020.113059. Epub 2020 Dec 3.
Eur J Med Chem. 2021.
PMID: 33310288
Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease.
Toublet FX, Lecoutey C, Lalut J, Hatat B, Davis A, Since M, Corvaisier S, Freret T, Sopkova de Oliveira Santos J, Claeysen S, Boulouard M, Dallemagne P, Rochais C.
Toublet FX, et al.
Molecules. 2019 Jul 31;24(15):2786. doi: 10.3390/molecules24152786.
Molecules. 2019.
PMID: 31370232
Free PMC article.
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In vivo emergence of rifampicin resistance by rpoB mutation in Listeria monocytogenes during therapy of prosthetic joint infection.
Isnard C, Fines-Guyon M, Toublet FX, Guerin F, Rogowski C, Vergnaud M, Cattoir V.
Isnard C, et al. Among authors: toublet fx.
Int J Antimicrob Agents. 2016 Nov;48(5):572-574. doi: 10.1016/j.ijantimicag.2016.07.016. Epub 2016 Sep 8.
Int J Antimicrob Agents. 2016.
PMID: 27659120
No abstract available.
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