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Monepantel is a non-competitive antagonist of nicotinic acetylcholine receptors from Ascaris suum and Oesophagostomum dentatum.
Int J Parasitol Drugs Drug Resist. 2018 Apr;8(1):36-42. doi: 10.1016/j.ijpddr.2017.12.001. Epub 2017 Dec 16.
Int J Parasitol Drugs Drug Resist. 2018.
PMID: 29366967
Free PMC article.
Pharmacological characterization of a homomeric nicotinic acetylcholine receptor formed by Ancylostoma caninum ACR-16.
Choudhary S, Tipton JG, Abongwa M, Brewer MT, Chelladurai JJ, Musselman N, Martin RJ, Robertson AP.
Choudhary S, et al. Among authors: tipton jg.
Invert Neurosci. 2019 Sep 5;19(4):11. doi: 10.1007/s10158-019-0231-0.
Invert Neurosci. 2019.
PMID: 31486912
Free PMC article.
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