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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2001 1
2002 18
2003 12
2004 10
2005 9
2006 7
2007 15
2008 10
2009 4
2010 4
2011 4
2012 1
2013 2
2014 1
2015 4
2016 2
2017 4
2018 6
2019 6
2020 6
2021 4
2022 8
2023 10
2024 5

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136 results

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Page 1
Discovery and optimization of narrow spectrum inhibitors of Tousled like kinase 2 (TLK2) using quantitative structure activity relationships.
Asquith CRM, East MP, Laitinen T, Alamillo-Ferrer C, Hartikainen E, Wells CI, Axtman AD, Drewry DH, Tizzard GJ, Poso A, Willson TM, Johnson GL. Asquith CRM, et al. Among authors: willson tm. Eur J Med Chem. 2024 Apr 2;271:116357. doi: 10.1016/j.ejmech.2024.116357. Online ahead of print. Eur J Med Chem. 2024. PMID: 38636130 Free article.
Discovery of a cell-active chikungunya virus nsP2 protease inhibitor using a covalent fragment-based screening approach.
Merten EM, Sears JD, Leisner TM, Hardy PB, Ghoshal A, Hossain MA, Asressu KH, Brown PJ, Stashko MA, Herring LE, Mordant AL, Webb TS, Mills CA, Barker NK, Arnold JJ, Cameron CE, Streblow DN, Moorman NJ, Heise M, Willson TM, Popov KI, Pearce KH. Merten EM, et al. Among authors: willson tm. bioRxiv [Preprint]. 2024 Mar 22:2024.03.22.586341. doi: 10.1101/2024.03.22.586341. bioRxiv. 2024. PMID: 38562906 Free PMC article. Preprint.
Discovery and Optimization of Narrow Spectrum Inhibitors of Tousled Like Kinase 2 (TLK2) Using Quantitative Structure Activity Relationships.
Asquith CRM, East MP, Laitinen T, Alamillo-Ferrer C, Hartikainen E, Wells CI, Axtman AD, Drewry DH, Tizzard GJ, Poso A, Willson TM, Johnson GL. Asquith CRM, et al. Among authors: willson tm. bioRxiv [Preprint]. 2023 Dec 28:2023.12.28.573261. doi: 10.1101/2023.12.28.573261. bioRxiv. 2023. PMID: 38234837 Free PMC article. Updated. Preprint.
Illuminating function of the understudied druggable kinome.
Gomez SM, Axtman AD, Willson TM, Major MB, Townsend RR, Sorger PK, Johnson GL. Gomez SM, et al. Among authors: willson tm. Drug Discov Today. 2024 Mar;29(3):103881. doi: 10.1016/j.drudis.2024.103881. Epub 2024 Jan 11. Drug Discov Today. 2024. PMID: 38218213 Review.
Fused Tetrahydroquinolines Are Interfering with Your Assay.
Bashore FM, Annor-Gyamfi J, Du Y, Katis V, Nwogbo F, Flax RG, Frye SV, Pearce KH, Fu H, Willson TM, Drewry DH, Axtman AD. Bashore FM, et al. Among authors: willson tm. J Med Chem. 2023 Nov 9;66(21):14434-14446. doi: 10.1021/acs.jmedchem.3c01277. Epub 2023 Oct 24. J Med Chem. 2023. PMID: 37874947 Free PMC article. Review.
136 results