Tikhomirov AS - Search Results

1

Synthesis and antitumor activity of cyclopentane-fused anthraquinone derivatives.

Tikhomirov AS, Sinkevich YB, Dezhenkova LG, Kaluzhny DN, Ilyinsky NS, Borshchevskiy VI, Schols D, Shchekotikhin AE. Tikhomirov AS, et al. Eur J Med Chem. 2024 Feb 5;265:116103. doi: 10.1016/j.ejmech.2023.116103. Epub 2023 Dec 30. Eur J Med Chem. 2024. PMID: 38176358

2

Thiadiazole-, selenadiazole- and triazole-fused anthraquinones as G-quadruplex targeting anticancer compounds.

Andreeva DV, Vedekhina TS, Gostev AS, Dezhenkova LG, Volodina YL, Markova AA, Nguyen MT, Ivanova OM, Dolgusheva VА, Varizhuk AM, Tikhomirov AS, Shchekotikhin AE. Andreeva DV, et al. Among authors: tikhomirov as. Eur J Med Chem. 2024 Mar 15;268:116222. doi: 10.1016/j.ejmech.2024.116222. Epub 2024 Feb 13. Eur J Med Chem. 2024. PMID: 38387333

3

Hybrid Molecules of Azithromycin with Chloramphenicol and Metronidazole: Synthesis and Study of Antibacterial Properties.

Volynkina IA, Bychkova EN, Karakchieva AO, Tikhomirov AS, Zatonsky GV, Solovieva SE, Martynov MM, Grammatikova NE, Tereshchenkov AG, Paleskava A, Konevega AL, Sergiev PV, Dontsova OA, Osterman IA, Shchekotikhin AE, Tevyashova AN. Volynkina IA, et al. Among authors: tikhomirov as. Pharmaceuticals (Basel). 2024 Jan 31;17(2):187. doi: 10.3390/ph17020187. Pharmaceuticals (Basel). 2024. PMID: 38399402 Free PMC article.

4

Water-soluble 4-(dimethylaminomethyl)heliomycin exerts greater antitumor effects than parental heliomycin by targeting the tNOX-SIRT1 axis and apoptosis in oral cancer cells.

Islam A, Chang YC, Chen XC, Weng CW, Chen CY, Wang CW, Chen MK, Tikhomirov AS, Shchekotikhin AE, Chueh PJ. Islam A, et al. Among authors: tikhomirov as. Elife. 2024 Apr 3;12:RP87873. doi: 10.7554/eLife.87873. Elife. 2024. PMID: 38567911 Free PMC article.

5

Design, Synthesis and In Vitro Investigation of Cabozantinib-Based PROTACs to Target c-Met Kinase.

Sachkova AA, Andreeva DV, Tikhomirov AS, Scherbakov AM, Salnikova DI, Sorokin DV, Bogdanov FB, Rysina YD, Shchekotikhin AE, Shchegravina ES, Fedorov AY. Sachkova AA, et al. Among authors: tikhomirov as. Pharmaceutics. 2022 Dec 16;14(12):2829. doi: 10.3390/pharmaceutics14122829. Pharmaceutics. 2022. PMID: 36559322 Free PMC article.

6

Computational and Biophysical Characterization of Heterocyclic Derivatives of Anthraquinone against Human Aurora Kinase A.

Singh M, Haque MA, Tikhomirov AS, Shchekotikhin AE, Das U, Kaur P. Singh M, et al. Among authors: tikhomirov as. ACS Omega. 2022 Oct 27;7(44):39603-39618. doi: 10.1021/acsomega.2c00740. eCollection 2022 Nov 8. ACS Omega. 2022. PMID: 36385832 Free PMC article.

7

Bis(chloroacetamidino)-Derived Heteroarene-Fused Anthraquinones Bind to and Cause Proteasomal Degradation of tNOX, Leading to c-Flip Downregulation and Apoptosis in Oral Cancer Cells.

Chang JS, Chen CY, Tikhomirov AS, Islam A, Liang RH, Weng CW, Wu WH, Shchekotikhin AE, Chueh PJ. Chang JS, et al. Among authors: tikhomirov as. Cancers (Basel). 2022 Sep 28;14(19):4719. doi: 10.3390/cancers14194719. Cancers (Basel). 2022. PMID: 36230644 Free PMC article.

8

Heterocyclic ring expansion yields anthraquinone derivatives potent against multidrug resistant tumor cells.

Tikhomirov AS, Tsvetkov VB, Volodina YL, Litvinova VA, Andreeva DV, Dezhenkova LG, Kaluzhny DN, Treshalin ID, Shtil AA, Shchekotikhin AE. Tikhomirov AS, et al. Bioorg Chem. 2022 Oct;127:105925. doi: 10.1016/j.bioorg.2022.105925. Epub 2022 Jun 4. Bioorg Chem. 2022. PMID: 35728293

9

Antibiotic heliomycin and its water-soluble 4-aminomethylated derivative provoke cell death in T24 bladder cancer cells by targeting sirtuin 1 (SIRT1).

Lin MH, Islam A, Liu YH, Weng CW, Zhan JH, Liang RH, Tikhomirov AS, Shchekotikhin AE, Chueh PJ. Lin MH, et al. Among authors: tikhomirov as. Am J Cancer Res. 2022 Mar 15;12(3):1042-1055. eCollection 2022. Am J Cancer Res. 2022. PMID: 35411221 Free PMC article.

10

Thiophene-2-carboxamide derivatives of anthraquinone: A new potent antitumor chemotype.

Volodina YL, Tikhomirov AS, Dezhenkova LG, Ramonova AA, Kononova AV, Andreeva DV, Kaluzhny DN, Schols D, Moisenovich MM, Shchekotikhin AE, Shtil AA. Volodina YL, et al. Among authors: tikhomirov as. Eur J Med Chem. 2021 Oct 5;221:113521. doi: 10.1016/j.ejmech.2021.113521. Epub 2021 May 24. Eur J Med Chem. 2021. PMID: 34082225

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