Thakur GA - Search Results

1

Negative allosteric modulation of CB₁ cannabinoid receptor signaling suppresses opioid-mediated reward.

Iyer V, Rangel-Barajas C, Woodward TJ, Kulkarni A, Cantwell L, Crystal JD, Mackie K, Rebec GV, Thakur GA, Hohmann AG. Iyer V, et al. Among authors: thakur ga. Pharmacol Res. 2022 Nov;185:106474. doi: 10.1016/j.phrs.2022.106474. Epub 2022 Sep 28. Pharmacol Res. 2022. PMID: 36179954 Free PMC article.

2

Selective activation of cannabinoid CB2 receptors suppresses neuropathic nociception induced by treatment with the chemotherapeutic agent paclitaxel in rats.

Rahn EJ, Zvonok AM, Thakur GA, Khanolkar AD, Makriyannis A, Hohmann AG. Rahn EJ, et al. Among authors: thakur ga. J Pharmacol Exp Ther. 2008 Nov;327(2):584-91. doi: 10.1124/jpet.108.141994. Epub 2008 Jul 29. J Pharmacol Exp Ther. 2008. PMID: 18664590 Free PMC article.

3

Pharmacological characterization of AM1710, a putative cannabinoid CB2 agonist from the cannabilactone class: antinociception without central nervous system side-effects.

Rahn EJ, Thakur GA, Wood JA, Zvonok AM, Makriyannis A, Hohmann AG. Rahn EJ, et al. Among authors: thakur ga. Pharmacol Biochem Behav. 2011 Jun;98(4):493-502. doi: 10.1016/j.pbb.2011.02.024. Epub 2011 Mar 5. Pharmacol Biochem Behav. 2011. PMID: 21382397 Free PMC article.

4

The maintenance of cisplatin- and paclitaxel-induced mechanical and cold allodynia is suppressed by cannabinoid CB₂ receptor activation and independent of CXCR4 signaling in models of chemotherapy-induced peripheral neuropathy.

Deng L, Guindon J, Vemuri VK, Thakur GA, White FA, Makriyannis A, Hohmann AG. Deng L, et al. Among authors: thakur ga. Mol Pain. 2012 Sep 22;8:71. doi: 10.1186/1744-8069-8-71. Mol Pain. 2012. PMID: 22998838 Free PMC article.

5

Expeditious synthesis, enantiomeric resolution, and enantiomer functional characterization of (4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): an allosteric agonist-positive allosteric modulator of α7 nicotinic acetylcholine receptors.

Thakur GA, Kulkarni AR, Deschamps JR, Papke RL. Thakur GA, et al. J Med Chem. 2013 Nov 14;56(21):8943-7. doi: 10.1021/jm401267t. Epub 2013 Oct 25. J Med Chem. 2013. PMID: 24090443 Free PMC article.

6

Microwave-assisted Expeditious and Efficient Synthesis of Cyclopentene Ring-fused Tetrahydroquinoline Derivatives Using Three-component Povarov Reaction.

Kulkarni AR, Thakur GA. Kulkarni AR, et al. Among authors: thakur ga. Tetrahedron Lett. 2013 Nov 27;54(48):10.1016/j.tetlet.2013.09.107. doi: 10.1016/j.tetlet.2013.09.107. Tetrahedron Lett. 2013. PMID: 24421568 Free PMC article.

7

Prophylactic cannabinoid administration blocks the development of paclitaxel-induced neuropathic nociception during analgesic treatment and following cessation of drug delivery.

Rahn EJ, Deng L, Thakur GA, Vemuri K, Zvonok AM, Lai YY, Makriyannis A, Hohmann AG. Rahn EJ, et al. Among authors: thakur ga. Mol Pain. 2014 Apr 18;10:27. doi: 10.1186/1744-8069-10-27. Mol Pain. 2014. PMID: 24742127 Free PMC article.

8

The analgesic-like properties of the alpha7 nAChR silent agonist NS6740 is associated with non-conducting conformations of the receptor.

Papke RL, Bagdas D, Kulkarni AR, Gould T, AlSharari SD, Thakur GA, Damaj MI. Papke RL, et al. Among authors: thakur ga. Neuropharmacology. 2015 Apr;91:34-42. doi: 10.1016/j.neuropharm.2014.12.002. Epub 2014 Dec 11. Neuropharmacology. 2015. PMID: 25497451 Free PMC article.

9

Small molecule inhibitors of PSD95-nNOS protein-protein interactions as novel analgesics.

Lee WH, Xu Z, Ashpole NM, Hudmon A, Kulkarni PM, Thakur GA, Lai YY, Hohmann AG. Lee WH, et al. Among authors: thakur ga. Neuropharmacology. 2015 Oct;97:464-75. doi: 10.1016/j.neuropharm.2015.05.038. Epub 2015 Jun 10. Neuropharmacology. 2015. PMID: 26071110 Free PMC article.

10

Novel Electrophilic and Photoaffinity Covalent Probes for Mapping the Cannabinoid 1 Receptor Allosteric Site(s).

Kulkarni PM, Kulkarni AR, Korde A, Tichkule RB, Laprairie RB, Denovan-Wright EM, Zhou H, Janero DR, Zvonok N, Makriyannis A, Cascio MG, Pertwee RG, Thakur GA. Kulkarni PM, et al. Among authors: thakur ga. J Med Chem. 2016 Jan 14;59(1):44-60. doi: 10.1021/acs.jmedchem.5b01303. Epub 2015 Nov 28. J Med Chem. 2016. PMID: 26529344 Free PMC article.

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