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Synthesis, biological evaluation and molecular modeling of benzofuran piperidine derivatives as Aβ antiaggregant.
Eur J Med Chem. 2021 Oct 15;222:113541. doi: 10.1016/j.ejmech.2021.113541. Epub 2021 May 25.
Eur J Med Chem. 2021.
PMID: 34116326
Structural optimization of pyrazolo[1,5-a]pyrimidine derivatives as potent and highly selective DPP-4 inhibitors.
Shen J, Deng X, Sun R, Tavallaie MS, Wang J, Cai Q, Lam C, Lei S, Fu L, Jiang F.
Shen J, et al. Among authors: tavallaie ms.
Eur J Med Chem. 2020 Dec 15;208:112850. doi: 10.1016/j.ejmech.2020.112850. Epub 2020 Sep 19.
Eur J Med Chem. 2020.
PMID: 32987315
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Surrogating and redirection of pyrazolo[1,5-a]pyrimidin-7(4H)-one core, a novel class of potent and selective DPP-4 inhibitors.
Deng X, Shen J, Zhu H, Xiao J, Sun R, Xie F, Lam C, Wang J, Qiao Y, Tavallaie MS, Hu Y, Du Y, Li J, Fu L, Jiang F.
Deng X, et al. Among authors: tavallaie ms.
Bioorg Med Chem. 2018 Feb 15;26(4):903-912. doi: 10.1016/j.bmc.2018.01.006. Epub 2018 Jan 10.
Bioorg Med Chem. 2018.
PMID: 29373269
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Anti-diabetic potential of Pueraria lobata root extract through promoting insulin signaling by PTP1B inhibition.
Sun R, Deng X, Zhang D, Xie F, Wang D, Wang J, Tavallaie MS, Jiang F, Fu L.
Sun R, et al. Among authors: tavallaie ms.
Bioorg Chem. 2019 Jun;87:12-15. doi: 10.1016/j.bioorg.2019.02.046. Epub 2019 Feb 22.
Bioorg Chem. 2019.
PMID: 30852232
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Identification of lipid-like salicylic acid-based derivatives as potent and membrane-permeable PTP1B inhibitors.
Li L, Tavallaie MS, Xie F, Xia Y, Liang Y, Jiang F, Fu L.
Li L, et al. Among authors: tavallaie ms.
Bioorg Chem. 2019 Dec;93:103296. doi: 10.1016/j.bioorg.2019.103296. Epub 2019 Sep 17.
Bioorg Chem. 2019.
PMID: 31585268
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Drug discovery approaches targeting the incretin pathway.
Deng X, Tavallaie MS, Sun R, Wang J, Cai Q, Shen J, Lei S, Fu L, Jiang F.
Deng X, et al. Among authors: tavallaie ms.
Bioorg Chem. 2020 Jun;99:103810. doi: 10.1016/j.bioorg.2020.103810. Epub 2020 Apr 2.
Bioorg Chem. 2020.
PMID: 32325333
Review.
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Moderation of mitochondrial respiration mitigates metabolic syndrome of aging.
Tavallaie M, Voshtani R, Deng X, Qiao Y, Jiang F, Collman JP, Fu L.
Tavallaie M, et al.
Proc Natl Acad Sci U S A. 2020 May 5;117(18):9840-9850. doi: 10.1073/pnas.1917948117. Epub 2020 Apr 17.
Proc Natl Acad Sci U S A. 2020.
PMID: 32303655
Free PMC article.
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Progranulin promotes melanoma progression by inhibiting natural killer cell recruitment to the tumor microenvironment.
Voshtani R, Song M, Wang H, Li X, Zhang W, Tavallaie MS, Yan W, Sun J, Wei F, Ma X.
Voshtani R, et al. Among authors: tavallaie ms.
Cancer Lett. 2019 Nov 28;465:24-35. doi: 10.1016/j.canlet.2019.08.018. Epub 2019 Sep 3.
Cancer Lett. 2019.
PMID: 31491449
Free PMC article.
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