Tapadar S - Search Results

1

A Novel Liver Cancer-Selective Histone Deacetylase Inhibitor Is Effective Against Hepatocellular Carcinoma and Induces Durable Responses with Immunotherapy.

Wu B, Tapadar S, Ruan Z, Sun CQ, Arnold RS, Olugbami JO, Johnston A, Arunsi U, Gaul DA, Petros JA, Kobayashi T, Duda DG, Oyelere AK. Wu B, et al. Among authors: tapadar s. bioRxiv [Preprint]. 2024 Mar 28:2024.03.27.587062. doi: 10.1101/2024.03.27.587062. bioRxiv. 2024. PMID: 38585757 Free PMC article. Preprint.

2

Isoxazole moiety in the linker region of HDAC inhibitors adjacent to the Zn-chelating group: effects on HDAC biology and antiproliferative activity.

Tapadar S, He R, Luchini DN, Billadeau DD, Kozikowski AP. Tapadar S, et al. Bioorg Med Chem Lett. 2009 Jun 1;19(11):3023-6. doi: 10.1016/j.bmcl.2009.04.058. Epub 2009 Apr 20. Bioorg Med Chem Lett. 2009. PMID: 19419863 Free PMC article.

3

Novel Selective Calpain 1 Inhibitors as Potential Therapeutics in Alzheimer's Disease.

Fà M, Zhang H, Staniszewski A, Saeed F, Shen LW, Schiefer IT, Siklos MI, Tapadar S, Litosh VA, Libien J, Petukhov PA, Teich AF, Thatcher GR, Arancio O. Fà M, et al. Among authors: tapadar s. J Alzheimers Dis. 2016;49(3):707-21. doi: 10.3233/JAD-150618. J Alzheimers Dis. 2016. PMID: 26484927 Free PMC article.

4

Design and synthesis of aryl ether inhibitors of the Bacillus anthracis enoyl-ACP reductase.

Tipparaju SK, Mulhearn DC, Klein GM, Chen Y, Tapadar S, Bishop MH, Yang S, Chen J, Ghassemi M, Santarsiero BD, Cook JL, Johlfs M, Mesecar AD, Johnson ME, Kozikowski AP. Tipparaju SK, et al. Among authors: tapadar s. ChemMedChem. 2008 Aug;3(8):1250-68. doi: 10.1002/cmdc.200800047. ChemMedChem. 2008. PMID: 18663709 Free PMC article.

5

Use of the nitrile oxide cycloaddition (NOC) reaction for molecular probe generation: a new class of enzyme selective histone deacetylase inhibitors (HDACIs) showing picomolar activity at HDAC6.

Kozikowski AP, Tapadar S, Luchini DN, Kim KH, Billadeau DD. Kozikowski AP, et al. Among authors: tapadar s. J Med Chem. 2008 Aug 14;51(15):4370-3. doi: 10.1021/jm8002894. Epub 2008 Jul 22. J Med Chem. 2008. PMID: 18642892 Free PMC article.

6

Exploiting translational stalling peptides in an effort to extend azithromycin interaction within the prokaryotic ribosome nascent peptide exit tunnel.

Washington AZ, Tapadar S, George A, Oyelere AK. Washington AZ, et al. Among authors: tapadar s. Bioorg Med Chem. 2015 Aug 15;23(16):5198-209. doi: 10.1016/j.bmc.2015.04.078. Epub 2015 May 6. Bioorg Med Chem. 2015. PMID: 26037612 Free PMC article.

7

A structure-activity relationship of non-peptide macrocyclic histone deacetylase inhibitors and their anti-proliferative and anti-inflammatory activities.

Tapadar S, Fathi S, Raji I, Omesiete W, Kornacki JR, Mwakwari SC, Miyata M, Mitsutake K, Li JD, Mrksich M, Oyelere AK. Tapadar S, et al. Bioorg Med Chem. 2015 Dec 15;23(24):7543-64. doi: 10.1016/j.bmc.2015.10.045. Epub 2015 Nov 2. Bioorg Med Chem. 2015. PMID: 26585275 Free PMC article.

8

Deferiprone: Pan-selective Histone Lysine Demethylase Inhibition Activity and Structure Activity Relationship Study.

Khodaverdian V, Tapadar S, MacDonald IA, Xu Y, Ho PY, Bridges A, Rajpurohit P, Sanghani BA, Fan Y, Thangaraju M, Hathaway NA, Oyelere AK. Khodaverdian V, et al. Among authors: tapadar s. Sci Rep. 2019 Mar 18;9(1):4802. doi: 10.1038/s41598-019-39214-1. Sci Rep. 2019. PMID: 30886160 Free PMC article.

9

Small Molecule Inhibitors Targeting Gα_i2 Protein Attenuate Migration of Cancer Cells.

Caggia S, Tapadar S, Wu B, Venugopal SV, Garrett AS, Kumar A, Stiffend JS, Davis JS, Oyelere AK, Khan SA. Caggia S, et al. Among authors: tapadar s. Cancers (Basel). 2020 Jun 19;12(6):1631. doi: 10.3390/cancers12061631. Cancers (Basel). 2020. PMID: 32575572 Free PMC article.

10

Liver-Targeting Class I Selective Histone Deacetylase Inhibitors Potently Suppress Hepatocellular Tumor Growth as Standalone Agents.

Tapadar S, Fathi S, Wu B, Sun CQ, Raji I, Moore SG, Arnold RS, Gaul DA, Petros JA, Oyelere AK. Tapadar S, et al. Cancers (Basel). 2020 Oct 23;12(11):3095. doi: 10.3390/cancers12113095. Cancers (Basel). 2020. PMID: 33114147 Free PMC article.

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