Szczepańska K - Search Results

1

Dual Piperidine-Based Histamine H₃ and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.

Szczepańska K, Karcz T, Dichiara M, Mogilski S, Kalinowska-Tłuścik J, Pilarski B, Leniak A, Pietruś W, Podlewska S, Popiołek-Barczyk K, Humphrys LJ, Ruiz-Cantero MC, Reiner-Link D, Leitzbach L, Łażewska D, Pockes S, Górka M, Zmysłowski A, Calmels T, Cobos EJ, Marrazzo A, Stark H, Bojarski AJ, Amata E, Kieć-Kononowicz K. Szczepańska K, et al. J Med Chem. 2023 Jul 27;66(14):9658-9683. doi: 10.1021/acs.jmedchem.3c00430. Epub 2023 Jul 7. J Med Chem. 2023. PMID: 37418295 Free PMC article.

2

Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands.

Szymańska E, Chałupnik P, Szczepańska K, Cuñado Moral AM, Pickering DS, Nielsen B, Johansen TN, Kieć-Kononowicz K. Szymańska E, et al. Among authors: szczepanska k. Bioorg Med Chem Lett. 2016 Nov 15;26(22):5568-5572. doi: 10.1016/j.bmcl.2016.09.075. Epub 2016 Sep 30. Bioorg Med Chem Lett. 2016. PMID: 27765511

3

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H₃R ligands.

Kuder KJ, Łażewska D, Kaleta M, Latacz G, Kottke T, Olejarz A, Karcz T, Fruziński A, Szczepańska K, Karolak-Wojciechowska J, Stark H, Kieć-Kononowicz K. Kuder KJ, et al. Among authors: szczepanska k. Bioorg Med Chem. 2017 May 15;25(10):2701-2712. doi: 10.1016/j.bmc.2017.03.031. Epub 2017 Mar 21. Bioorg Med Chem. 2017. PMID: 28372935

4

Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors.

Szymańska E, Nielsen B, Johansen TN, Cuñado Moral AM, Pickering DS, Szczepańska K, Mickowska A, Kieć-Kononowicz K. Szymańska E, et al. Among authors: szczepanska k. Eur J Med Chem. 2017 Sep 29;138:874-883. doi: 10.1016/j.ejmech.2017.07.007. Epub 2017 Jul 8. Eur J Med Chem. 2017. PMID: 28738307

5

Histamine H3 Receptor Ligands in the Group of (Homo)piperazine Derivatives.

Szczepanska K, Kuder K, Kiec-Kononowicz K. Szczepanska K, et al. Curr Med Chem. 2018;25(14):1609-1626. doi: 10.2174/0929867325666171123203550. Curr Med Chem. 2018. PMID: 29173145 Review.

6

Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H₃R ligands.

Szczepańska K, Karcz T, Mogilski S, Siwek A, Kuder KJ, Latacz G, Kubacka M, Hagenow S, Lubelska A, Olejarz A, Kotańska M, Sadek B, Stark H, Kieć-Kononowicz K. Szczepańska K, et al. Eur J Med Chem. 2018 May 25;152:223-234. doi: 10.1016/j.ejmech.2018.04.043. Epub 2018 Apr 25. Eur J Med Chem. 2018. PMID: 29723785

7

The histamine H₃ receptor inverse agonist pitolisant reduces body weight in obese mice.

Kotańska M, Kuder KJ, Szczepańska K, Sapa J, Kieć-Kononowicz K. Kotańska M, et al. Among authors: szczepanska k. Naunyn Schmiedebergs Arch Pharmacol. 2018 Aug;391(8):875-881. doi: 10.1007/s00210-018-1516-2. Epub 2018 May 25. Naunyn Schmiedebergs Arch Pharmacol. 2018. PMID: 29802412 Free PMC article.

8

Optimization and preclinical evaluation of novel histamine H₃receptor ligands: Acetyl and propionyl phenoxyalkyl piperazine derivatives.

Szczepańska K, Karcz T, Kotańska M, Siwek A, Kuder KJ, Latacz G, Mogilski S, Hagenow S, Lubelska A, Sobolewski M, Stark H, Kieć-Kononowicz K. Szczepańska K, et al. Bioorg Med Chem. 2018 Dec 15;26(23-24):6056-6066. doi: 10.1016/j.bmc.2018.11.010. Epub 2018 Nov 10. Bioorg Med Chem. 2018. PMID: 30448256

9

KSK19 - Novel histamine H3 receptor ligand reduces body weight in diet induced obese mice.

Kotańska M, Mika K, Reguła K, Szczepańska K, Szafarz M, Bednarski M, Olejarz-Maciej A, Nowak K, Latacz G, Mogilski S, Kuder KJ, Kieć-Kononowicz K, Sapa J. Kotańska M, et al. Among authors: szczepanska k. Biochem Pharmacol. 2019 Oct;168:193-203. doi: 10.1016/j.bcp.2019.07.006. Epub 2019 Jul 8. Biochem Pharmacol. 2019. PMID: 31295465

10

Structural modifications and in vitro pharmacological evaluation of 4-pyridyl-piperazine derivatives as an active and selective histamine H₃ receptor ligands.

Szczepańska K, Karcz T, Siwek A, Kuder KJ, Latacz G, Bednarski M, Szafarz M, Hagenow S, Lubelska A, Olejarz-Maciej A, Sobolewski M, Mika K, Kotańska M, Stark H, Kieć-Kononowicz K. Szczepańska K, et al. Bioorg Chem. 2019 Oct;91:103071. doi: 10.1016/j.bioorg.2019.103071. Epub 2019 Jun 20. Bioorg Chem. 2019. PMID: 31362197

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