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Structure-Based Discovery of a New Selectivity-Enabling Motif for the FK506-Binding Protein 51.
J Med Chem. 2023 Apr 27;66(8):5965-5980. doi: 10.1021/acs.jmedchem.3c00249. Epub 2023 Apr 14.
J Med Chem. 2023.
PMID: 37058391
Structure-Based Design of High-Affinity Macrocyclic FKBP51 Inhibitors.
Bauder M, Meyners C, Purder PL, Merz S, Sugiarto WO, Voll AM, Heymann T, Hausch F.
Bauder M, et al. Among authors: sugiarto wo.
J Med Chem. 2021 Mar 25;64(6):3320-3349. doi: 10.1021/acs.jmedchem.0c02195. Epub 2021 Mar 5.
J Med Chem. 2021.
PMID: 33666419
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Deconstructing Protein Binding of Sulfonamides and Sulfonamide Analogues.
Purder PL, Meyners C, Sugiarto WO, Kolos J, Löhr F, Gebel J, Nehls T, Dötsch V, Lermyte F, Hausch F.
Purder PL, et al. Among authors: sugiarto wo.
JACS Au. 2023 Aug 25;3(9):2478-2486. doi: 10.1021/jacsau.3c00241. eCollection 2023 Sep 25.
JACS Au. 2023.
PMID: 37772190
Free PMC article.
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Synthesis and structure activity relationship of 1, 3-benzo-thiazine-2-thiones as selective HDAC8 inhibitors.
Wolff B, Jänsch N, Sugiarto WO, Frühschulz S, Lang M, Altintas R, Oehme I, Meyer-Almes FJ.
Wolff B, et al. Among authors: sugiarto wo.
Eur J Med Chem. 2019 Dec 15;184:111756. doi: 10.1016/j.ejmech.2019.111756. Epub 2019 Oct 7.
Eur J Med Chem. 2019.
PMID: 31630054
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Kinetically selective and potent inhibitors of HDAC8.
Schweipert M, Jänsch N, Sugiarto WO, Meyer-Almes FJ.
Schweipert M, et al. Among authors: sugiarto wo.
Biol Chem. 2019 May 27;400(6):733-743. doi: 10.1515/hsz-2018-0363.
Biol Chem. 2019.
PMID: 30521473
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Discovery of a Potent Proteolysis Targeting Chimera Enables Targeting the Scaffolding Functions of FK506-Binding Protein 51 (FKBP51).
Geiger TM, Walz M, Meyners C, Kuehn A, Dreizler JK, Sugiarto WO, Maciel EVS, Zheng M, Lermyte F, Hausch F.
Geiger TM, et al. Among authors: sugiarto wo.
Angew Chem Int Ed Engl. 2024 Jan 15;63(3):e202309706. doi: 10.1002/anie.202309706. Epub 2023 Dec 14.
Angew Chem Int Ed Engl. 2024.
PMID: 37942685
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Switching the Switch: Ligand Induced Disulfide Formation in HDAC8.
Jänsch N, Sugiarto WO, Muth M, Kopranovic A, Desczyk C, Ballweg M, Kirschhöfer F, Brenner-Weiss G, Meyer-Almes FJ.
Jänsch N, et al. Among authors: sugiarto wo.
Chemistry. 2020 Oct 15;26(58):13249-13255. doi: 10.1002/chem.202001712. Epub 2020 Sep 11.
Chemistry. 2020.
PMID: 32428298
Free PMC article.
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