Steinmetzer T - Search Results

1

Acylated 1H-1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action.

Korff M, Imberg L, Will JM, Bückreiß N, Kalinina SA, Wenzel BM, Kastner GA, Daniliuc CG, Barth M, Ovsepyan RA, Butov KR, Humpf HU, Lehr M, Panteleev MA, Poso A, Karst U, Steinmetzer T, Bendas G, Kalinin DV. Korff M, et al. Among authors: steinmetzer t. J Med Chem. 2020 Nov 12;63(21):13159-13186. doi: 10.1021/acs.jmedchem.0c01635. Epub 2020 Oct 22. J Med Chem. 2020. PMID: 33089691

2

Progress in the development of synthetic thrombin inhibitors as new orally active anticoagulants.

Steinmetzer T, Stürzebecher J. Steinmetzer T, et al. Curr Med Chem. 2004 Sep;11(17):2297-321. doi: 10.2174/0929867043364540. Curr Med Chem. 2004. PMID: 15379714 Review.

3

New substrate analogue inhibitors of factor Xa containing 4-amidinobenzylamide as P1 residue: part 1.

Schweinitz A, Stürzebecher A, Stürzebecher U, Schuster O, Stürzebecher J, Steinmetzer T. Schweinitz A, et al. Among authors: steinmetzer t. Med Chem. 2006 Jul;2(4):349-61. doi: 10.2174/157340606777724040. Med Chem. 2006. PMID: 16848746

4

From selective substrate analogue factor Xa inhibitors to dual inhibitors of thrombin and factor Xa. Part 3.

Dönnecke D, Schweinitz A, Stürzebecher A, Steinmetzer P, Schuster M, Stürzebecher U, Nicklisch S, Stürzebecher J, Steinmetzer T. Dönnecke D, et al. Among authors: steinmetzer t, steinmetzer p. Bioorg Med Chem Lett. 2007 Jun 15;17(12):3322-9. doi: 10.1016/j.bmcl.2007.03.105. Epub 2007 Apr 6. Bioorg Med Chem Lett. 2007. PMID: 17462889

5

Modification of the N-terminal sulfonyl residue in 3-amidinophenylalanine-based matriptase inhibitors.

Steinmetzer T, Dönnecke D, Korsonewski M, Neuwirth C, Steinmetzer P, Schulze A, Saupe SM, Schweinitz A. Steinmetzer T, et al. Among authors: steinmetzer p. Bioorg Med Chem Lett. 2009 Jan 1;19(1):67-73. doi: 10.1016/j.bmcl.2008.11.019. Epub 2008 Nov 13. Bioorg Med Chem Lett. 2009. PMID: 19036586

6

Potent inhibitors of furin and furin-like proprotein convertases containing decarboxylated P1 arginine mimetics.

Becker GL, Sielaff F, Than ME, Lindberg I, Routhier S, Day R, Lu Y, Garten W, Steinmetzer T. Becker GL, et al. Among authors: steinmetzer t. J Med Chem. 2010 Feb 11;53(3):1067-75. doi: 10.1021/jm9012455. J Med Chem. 2010. PMID: 20038105 Free PMC article.

7

Identification of the first low-molecular-weight inhibitors of matriptase-2.

Sisay MT, Steinmetzer T, Stirnberg M, Maurer E, Hammami M, Bajorath J, Gütschow M. Sisay MT, et al. Among authors: steinmetzer t. J Med Chem. 2010 Aug 12;53(15):5523-35. doi: 10.1021/jm100183e. J Med Chem. 2010. PMID: 20684597

8

New furin inhibitors based on weakly basic amidinohydrazones.

Sielaff F, Than ME, Bevec D, Lindberg I, Steinmetzer T. Sielaff F, et al. Among authors: steinmetzer t. Bioorg Med Chem Lett. 2011 Jan 15;21(2):836-40. doi: 10.1016/j.bmcl.2010.11.092. Epub 2010 Nov 25. Bioorg Med Chem Lett. 2011. PMID: 21168329 Free PMC article.

9

Development of substrate analogue inhibitors for the human airway trypsin-like protease HAT.

Sielaff F, Böttcher-Friebertshäuser E, Meyer D, Saupe SM, Volk IM, Garten W, Steinmetzer T. Sielaff F, et al. Among authors: steinmetzer t. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4860-4. doi: 10.1016/j.bmcl.2011.06.033. Epub 2011 Jun 21. Bioorg Med Chem Lett. 2011. PMID: 21741839

10

New substrate analogue furin inhibitors derived from 4-amidinobenzylamide.

Becker GL, Hardes K, Steinmetzer T. Becker GL, et al. Among authors: steinmetzer t. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4695-7. doi: 10.1016/j.bmcl.2011.06.091. Epub 2011 Jun 25. Bioorg Med Chem Lett. 2011. PMID: 21757345

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