Stapleton P - Search Results

1

Regioselective glycosylation of novobiocin alters activity.

Sun G, de Resende PE, Stapleton P, Kuta M, Wang X, Haider S, Yang M. Sun G, et al. Among authors: stapleton p. Carbohydr Res. 2017 Nov 27;452:116-121. doi: 10.1016/j.carres.2017.10.011. Epub 2017 Oct 22. Carbohydr Res. 2017. PMID: 29096184

2

High throughput discovery of heteroaromatic-modifying enzymes allows enhancement of novobiocin selectivity.

Patel SM, de la Fuente M, Ke S, Guimarães AM, Oliyide AO, Ji X, Stapleton P, Osbourn A, Pan Y, Bowles DJ, Davis BG, Schatzlein A, Yang M. Patel SM, et al. Among authors: stapleton p. Chem Commun (Camb). 2011 Oct 14;47(38):10569-71. doi: 10.1039/c1cc13552j. Epub 2011 Aug 24. Chem Commun (Camb). 2011. PMID: 21863200

3

Boronic acid inhibitors of the class A β-lactamase KPC-2.

Zhou J, Stapleton P, Haider S, Healy J. Zhou J, et al. Among authors: stapleton p. Bioorg Med Chem. 2018 Jul 15;26(11):2921-2927. doi: 10.1016/j.bmc.2018.04.055. Epub 2018 Apr 27. Bioorg Med Chem. 2018. PMID: 29784271

4

Synthesis and in Silico Modelling of the Potential Dual Mechanistic Activity of Small Cationic Peptides Potentiating the Antibiotic Novobiocin against Susceptible and Multi-Drug Resistant Escherichia coli.

Passarini I, Resende PE, Soares S, Tahmasi T, Stapleton P, Malkinson J, Zloh M, Rossiter S. Passarini I, et al. Among authors: stapleton p. Int J Mol Sci. 2020 Nov 30;21(23):9134. doi: 10.3390/ijms21239134. Int J Mol Sci. 2020. PMID: 33266278 Free PMC article.

5

Triazole-substituted phenylboronic acids as tunable lead inhibitors of KPC-2 antibiotic resistance.

Zhou J, Stapleton P, Xavier-Junior FH, Schatzlein A, Haider S, Healy J, Wells G. Zhou J, et al. Among authors: stapleton p. Eur J Med Chem. 2022 Oct 5;240:114571. doi: 10.1016/j.ejmech.2022.114571. Epub 2022 Jun 28. Eur J Med Chem. 2022. PMID: 35792385 Free article.

6

LY2183240 regioisomers act as competitive and selective inhibitors of class C β-lactamases.

de Resende PE, Soares S, Zloh M, Gibbons S, Stapleton P. de Resende PE, et al. Among authors: stapleton p. Int J Antimicrob Agents. 2023 May;61(5):106774. doi: 10.1016/j.ijantimicag.2023.106774. Epub 2023 Mar 7. Int J Antimicrob Agents. 2023. PMID: 36893812

7

Antibacterial acylphloroglucinols from Hypericum olympicum.

Shiu WK, Rahman MM, Curry J, Stapleton P, Zloh M, Malkinson JP, Gibbons S. Shiu WK, et al. Among authors: stapleton p. J Nat Prod. 2012 Mar 23;75(3):336-43. doi: 10.1021/np2003319. Epub 2011 Sep 7. J Nat Prod. 2012. PMID: 21899267

8

In Vitro Antibacterial Activity of Prenylated Guanidine Alkaloids from Pterogyne nitens and Synthetic Analogues.

Coqueiro A, Regasini LO, Stapleton P, da Silva Bolzani V, Gibbons S. Coqueiro A, et al. Among authors: stapleton p. J Nat Prod. 2014 Aug 22;77(8):1972-5. doi: 10.1021/np500281c. Epub 2014 Aug 4. J Nat Prod. 2014. PMID: 25089583

9

Antistaphylococcal Prenylated Acylphoroglucinol and Xanthones from Kielmeyera variabilis.

Coqueiro A, Choi YH, Verpoorte R, Gupta KB, De Mieri M, Hamburger M, Young MC, Stapleton P, Gibbons S, Bolzani Vda S. Coqueiro A, et al. Among authors: stapleton p. J Nat Prod. 2016 Mar 25;79(3):470-6. doi: 10.1021/acs.jnatprod.5b00858. Epub 2016 Feb 22. J Nat Prod. 2016. PMID: 26900954

10

A New Era of Pulmonary Delivery of Nano-antimicrobial Therapeutics to Treat Chronic Pulmonary Infections.

Merchant Z, Buckton G, Taylor KM, Stapleton P, Saleem IY, Zariwala MG, Somavarapu S. Merchant Z, et al. Among authors: stapleton p. Curr Pharm Des. 2016;22(17):2577-98. doi: 10.2174/1381612822666160317142139. Curr Pharm Des. 2016. PMID: 26983671 Review.

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