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Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: a novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives.
Ranise A, Spallarossa A, Schenone S, Bruno O, Bondavalli F, Vargiu L, Marceddu T, Mura M, La Colla P, Pani A. Ranise A, et al. Among authors: spallarossa a. J Med Chem. 2003 Feb 27;46(5):768-81. doi: 10.1021/jm0209984. J Med Chem. 2003. PMID: 12593657
Synthesis and antiproliferative activity of basic thioanalogues of merbarone.
Ranise A, Spallarossa A, Schenone S, Bruno O, Bondavalli F, Pani A, Marongiu ME, Mascia V, La Colla P, Loddo R. Ranise A, et al. Among authors: spallarossa a. Bioorg Med Chem. 2003 Jun 12;11(12):2575-89. doi: 10.1016/s0968-0896(03)00158-5. Bioorg Med Chem. 2003. PMID: 12757725
Synthesis of N-substituted-N-acylthioureas of 4-substituted piperazines endowed with local anaesthetic, antihyperlipidemic, antiproliferative activities and antiarrythmic, analgesic, antiaggregating actions.
Ranise A, Spallarossa A, Bruno O, Schenone S, Fossa P, Menozzi G, Bondavalli F, Mosti L, Capuano A, Mazzeo F, Falcone G, Filippelli W. Ranise A, et al. Among authors: spallarossa a. Farmaco. 2003 Sep;58(9):765-80. doi: 10.1016/S0014-827X(03)00132-0. Farmaco. 2003. PMID: 13679169
Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives.
Ranise A, Spallarossa A, Cesarini S, Bondavalli F, Schenone S, Bruno O, Menozzi G, Fossa P, Mosti L, La Colla M, Sanna G, Murreddu M, Collu G, Busonera B, Marongiu ME, Pani A, La Colla P, Loddo R. Ranise A, et al. Among authors: spallarossa a. J Med Chem. 2005 Jun 2;48(11):3858-73. doi: 10.1021/jm049252r. J Med Chem. 2005. PMID: 15916438
Identification of a novel pyrazolo[3,4-d]pyrimidine able to inhibit cell proliferation of a human osteogenic sarcoma in vitro and in a xenograft model in mice.
Manetti F, Santucci A, Locatelli GA, Maga G, Spreafico A, Serchi T, Orlandini M, Bernardini G, Caradonna NP, Spallarossa A, Brullo C, Schenone S, Bruno O, Ranise A, Bondavalli F, Hoffmann O, Bologna M, Angelucci A, Botta M. Manetti F, et al. Among authors: spallarossa a. J Med Chem. 2007 Nov 15;50(23):5579-88. doi: 10.1021/jm061449r. Epub 2007 Oct 11. J Med Chem. 2007. PMID: 17929792
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate.
Cesarini S, Spallarossa A, Ranise A, Bruno O, La Colla P, Secci B, Collu G, Loddo R. Cesarini S, et al. Among authors: spallarossa a. Bioorg Med Chem. 2008 Apr 1;16(7):4173-85. doi: 10.1016/j.bmc.2007.12.046. Epub 2007 Dec 25. Bioorg Med Chem. 2008. PMID: 18226533
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Cesarini S, Spallarossa A, Ranise A, Schenone S, Bruno O, La Colla P, Casula L, Collu G, Sanna G, Loddo R. Cesarini S, et al. Among authors: spallarossa a. Bioorg Med Chem. 2008 Jun 15;16(12):6353-63. doi: 10.1016/j.bmc.2008.05.010. Epub 2008 May 7. Bioorg Med Chem. 2008. PMID: 18502646
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Spallarossa A, Cesarini S, Ranise A, Schenone S, Bruno O, Borassi A, La Colla P, Pezzullo M, Sanna G, Collu G, Secci B, Loddo R. Spallarossa A, et al. Eur J Med Chem. 2009 May;44(5):2190-201. doi: 10.1016/j.ejmech.2008.10.032. Epub 2008 Nov 5. Eur J Med Chem. 2009. PMID: 19058881
65 results