Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
4 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models.
Proc Natl Acad Sci U S A. 2023 Jan 3;120(1):e2211297120. doi: 10.1073/pnas.2211297120. Epub 2022 Dec 27.
Proc Natl Acad Sci U S A. 2023.
PMID: 36574664
Free PMC article.
Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based Optimization.
Teuscher KB, Meyers KM, Wei Q, Mills JJ, Tian J, Alvarado J, Sai J, Van Meveren M, South TM, Rietz TA, Zhao B, Moore WJ, Stott GM, Tansey WP, Lee T, Fesik SW.
Teuscher KB, et al. Among authors: south tm.
J Med Chem. 2022 Apr 28;65(8):6287-6312. doi: 10.1021/acs.jmedchem.2c00195. Epub 2022 Apr 18.
J Med Chem. 2022.
PMID: 35436124
Free PMC article.
Item in Clipboard
Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors.
Teuscher KB, Mills JJ, Tian J, Han C, Meyers KM, Sai J, South TM, Crow MM, Van Meveren M, Sensintaffar JL, Zhao B, Amporndanai K, Moore WJ, Stott GM, Tansey WP, Lee T, Fesik SW.
Teuscher KB, et al. Among authors: south tm.
J Med Chem. 2023 Dec 28;66(24):16783-16806. doi: 10.1021/acs.jmedchem.3c01529. Epub 2023 Dec 12.
J Med Chem. 2023.
PMID: 38085679
Item in Clipboard
Using NMR Spectroscopy To Measure Protein Binding Capacity on Gold Nanoparticles.
Perera YR, South TM, Hughes AC, Parkhurst AN, Williams OC, Davidson MB, Wilks CA, Mlsna DA, Fitzkee NC.
Perera YR, et al. Among authors: south tm.
J Chem Educ. 2020 Mar 10;97(3):820-824. doi: 10.1021/acs.jchemed.9b00625. Epub 2020 Jan 21.
J Chem Educ. 2020.
PMID: 34045774
Free PMC article.
Item in Clipboard
Cite
Cite