Sopkova de Oliveira Santos J - Search Results

1

Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease.

Toublet FX, Lecoutey C, Lalut J, Hatat B, Davis A, Since M, Corvaisier S, Freret T, Sopkova de Oliveira Santos J, Claeysen S, Boulouard M, Dallemagne P, Rochais C. Toublet FX, et al. Among authors: sopkova de oliveira santos j. Molecules. 2019 Jul 31;24(15):2786. doi: 10.3390/molecules24152786. Molecules. 2019. PMID: 31370232 Free PMC article.

2

3D-QSAR and docking studies of selective GSK-3beta inhibitors. Comparison with a thieno[2,3-b]pyrrolizinone derivative, a new potential lead for GSK-3beta ligands.

Lescot E, Bureau R, Sopkova-de Oliveira Santos J, Rochais C, Lisowski V, Lancelot JC, Rault S. Lescot E, et al. Among authors: sopkova de oliveira santos j. J Chem Inf Model. 2005 May-Jun;45(3):708-15. doi: 10.1021/ci050008y. J Chem Inf Model. 2005. PMID: 15921460

3

Synthesis of new dipyrrolo- and furopyrrolopyrazinones related to tripentones and their biological evaluation as potential kinases (CDKs1-5, GSK-3) inhibitors.

Rochais C, Duc NV, Lescot E, Sopkova-de Oliveira Santos J, Bureau R, Meijer L, Dallemagne P, Rault S. Rochais C, et al. Among authors: sopkova de oliveira santos j. Eur J Med Chem. 2009 Feb;44(2):708-16. doi: 10.1016/j.ejmech.2008.05.011. Epub 2008 May 23. Eur J Med Chem. 2009. PMID: 18586356

4

Synthesis and biological evaluation of new donepezil-like Thiaindanones as AChE inhibitors.

Omran Z, Stiebing S, Godard AM, Sopkova-De Oliveira-Santos J, Dallemagne P. Omran Z, et al. Among authors: sopkova de oliveira santos j. J Enzyme Inhib Med Chem. 2008 Oct;23(5):696-703. doi: 10.1080/14756360802208053. J Enzyme Inhib Med Chem. 2008. PMID: 18821258

5

Hydrogenative desulphurization of thienopyrrolizinones: an easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity.

Perri V, Rochais C, Sopkova-de Oliveira Santos J, Legay R, Cresteil T, Dallemagne P, Rault S. Perri V, et al. Among authors: sopkova de oliveira santos j. Eur J Med Chem. 2010 Mar;45(3):1146-50. doi: 10.1016/j.ejmech.2009.12.021. Epub 2009 Dec 21. Eur J Med Chem. 2010. PMID: 20053482

6

Virtual screening discovery of new acetylcholinesterase inhibitors issued from CERMN chemical library.

Sopkova-de Oliveira Santos J, Lesnard A, Agondanou JH, Dupont N, Godard AM, Stiebing S, Rochais C, Fabis F, Dallemagne P, Bureau R, Rault S. Sopkova-de Oliveira Santos J, et al. J Chem Inf Model. 2010 Mar 22;50(3):422-8. doi: 10.1021/ci900491t. J Chem Inf Model. 2010. PMID: 20196555

7

Interpretation of honeybees contact toxicity associated to acetylcholinesterase inhibitors.

Dulin F, Halm-Lemeille MP, Lozano S, Lepailleur A, Sopkova-de Oliveira Santos J, Rault S, Bureau R. Dulin F, et al. Among authors: sopkova de oliveira santos j. Ecotoxicol Environ Saf. 2012 May;79:13-21. doi: 10.1016/j.ecoenv.2012.01.007. Epub 2012 Feb 8. Ecotoxicol Environ Saf. 2012. PMID: 22321412

8

New hypotheses for the binding mode of 4- and 7-substituted indazoles in the active site of neuronal nitric oxide synthase.

Lohou E, Sopkova-de Oliveira Santos J, Schumann-Bard P, Boulouard M, Stiebing S, Rault S, Collot V. Lohou E, et al. Among authors: sopkova de oliveira santos j. Bioorg Med Chem. 2012 Sep 1;20(17):5296-304. doi: 10.1016/j.bmc.2012.06.025. Epub 2012 Jul 3. Bioorg Med Chem. 2012. PMID: 22831803

9

Novel multitarget-directed ligands (MTDLs) with acetylcholinesterase (AChE) inhibitory and serotonergic subtype 4 receptor (5-HT4R) agonist activities as potential agents against Alzheimer's disease: the design of donecopride.

Rochais C, Lecoutey C, Gaven F, Giannoni P, Hamidouche K, Hedou D, Dubost E, Genest D, Yahiaoui S, Freret T, Bouet V, Dauphin F, Sopkova de Oliveira Santos J, Ballandonne C, Corvaisier S, Malzert-Fréon A, Legay R, Boulouard M, Claeysen S, Dallemagne P. Rochais C, et al. Among authors: sopkova de oliveira santos j. J Med Chem. 2015 Apr 9;58(7):3172-87. doi: 10.1021/acs.jmedchem.5b00115. Epub 2015 Mar 31. J Med Chem. 2015. PMID: 25793650 Free article.

10

Novel benzylidenephenylpyrrolizinones with pleiotropic activities potentially useful in Alzheimer's disease treatment.

Jourdan JP, Since M, El Kihel L, Lecoutey C, Corvaisier S, Legay R, Sopkova-de Oliveira Santos J, Cresteil T, Malzert-Fréon A, Rochais C, Dallemagne P. Jourdan JP, et al. Among authors: sopkova de oliveira santos j. Eur J Med Chem. 2016 May 23;114:365-79. doi: 10.1016/j.ejmech.2016.03.023. Epub 2016 Mar 12. Eur J Med Chem. 2016. PMID: 27046230

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