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9-Azido-9-deoxy-2,3-difluorosialic Acid as a Subnanomolar Inhibitor against Bacterial Sialidases.
J Org Chem. 2019 Jun 7;84(11):6697-6708. doi: 10.1021/acs.joc.9b00385. Epub 2019 May 24.
J Org Chem. 2019.
PMID: 31083938
Free PMC article.
Streptococcus pneumoniae Sialidase SpNanB-Catalyzed One-Pot Multienzyme (OPME) Synthesis of 2,7-Anhydro-Sialic Acids as Selective Sialidase Inhibitors.
Xiao A, Slack TJ, Li Y, Shi D, Yu H, Li W, Liu Y, Chen X.
Xiao A, et al. Among authors: slack tj.
J Org Chem. 2018 Sep 21;83(18):10798-10804. doi: 10.1021/acs.joc.8b01519. Epub 2018 Aug 23.
J Org Chem. 2018.
PMID: 30105908
Free PMC article.
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Triazole-linked transition state analogs as selective inhibitors against V. cholerae sialidase.
Slack TJ, Li W, Shi D, McArthur JB, Zhao G, Li Y, Xiao A, Khedri Z, Yu H, Liu Y, Chen X.
Slack TJ, et al.
Bioorg Med Chem. 2018 Nov 15;26(21):5751-5757. doi: 10.1016/j.bmc.2018.10.028. Epub 2018 Oct 27.
Bioorg Med Chem. 2018.
PMID: 30389408
Free PMC article.
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Highly efficient chemoenzymatic synthesis and facile purification of α-Gal pentasaccharyl ceramide Galα3nLc4βCer.
Santra A, Li Y, Yu H, Slack TJ, Wang PG, Chen X.
Santra A, et al. Among authors: slack tj.
Chem Commun (Camb). 2017 Jul 20;53(59):8280-8283. doi: 10.1039/c7cc04090c.
Chem Commun (Camb). 2017.
PMID: 28695219
Free PMC article.
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Local Mechanical Perturbation Provides an Effective Means to Regulate the Growth and Assembly of Functional Peptide Fibrils.
Karsai A, Slack TJ, Malekan H, Khoury F, Lin WF, Tran V, Cox D, Toney M, Chen X, Liu GY.
Karsai A, et al. Among authors: slack tj.
Small. 2016 Dec;12(46):6407-6415. doi: 10.1002/smll.201601657. Epub 2016 Sep 30.
Small. 2016.
PMID: 27689936
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