Silvestri R - Search Results

1

Targeting the Grb2 cSH3 domain: Design, synthesis and biological evaluation of the first series of modulators.

Bufano M, Puxeddu M, Nalli M, La Regina G, Toto A, Liberati FR, Paone A, Cutruzzolà F, Masci D, Bigogno C, Dondio G, Silvestri R, Gianni S, Coluccia A. Bufano M, et al. Among authors: silvestri r. Bioorg Chem. 2023 Sep;138:106607. doi: 10.1016/j.bioorg.2023.106607. Epub 2023 May 11. Bioorg Chem. 2023. PMID: 37210829 Free article.

2

Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors.

Silvestri R, Artico M, De Martino G, Novellino E, Greco G, Lavecchia A, Massa S, Loi AG, Doratiotto S, La Colla P. Silvestri R, et al. Bioorg Med Chem. 2000 Sep;8(9):2305-9. doi: 10.1016/s0968-0896(00)00144-9. Bioorg Med Chem. 2000. PMID: 11026542

3

Simple, potent, and selective pyrrole inhibitors of monoamine oxidase types A and B.

Silvestri R, La Regina G, De Martino G, Artico M, Befani O, Palumbo M, Agostinelli E, Turini P. Silvestri R, et al. J Med Chem. 2003 Mar 13;46(6):917-20. doi: 10.1021/jm0256124. J Med Chem. 2003. PMID: 12620068

4

Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: synthesis and SAR studies.

Silvestri R, De Martino G, La Regina G, Artico M, Massa S, Vargiu L, Mura M, Loi AG, Marceddu T, La Colla P. Silvestri R, et al. J Med Chem. 2003 Jun 5;46(12):2482-93. doi: 10.1021/jm0211063. J Med Chem. 2003. PMID: 12773052

5

Anti-HIV-1 activity of pyrryl aryl sulfone (PAS) derivatives: synthesis and SAR studies of novel esters and amides at the position 2 of the pyrrole nucleus.

Silvestri R, Artico M, La Regina G, De Martino G, La Colla M, Loddo R, La Colla P. Silvestri R, et al. Farmaco. 2004 Mar;59(3):201-10. doi: 10.1016/j.farmac.2003.11.004. Farmaco. 2004. PMID: 14987983

6

Simple, short peptide derivatives of a sulfonylindolecarboxamide (L-737,126) active in vitro against HIV-1 wild type and variants carrying non-nucleoside reverse transcriptase inhibitor resistance mutations.

Silvestri R, Artico M, De Martino G, La Regina G, Loddo R, La Colla M, Mura M, La Colla P. Silvestri R, et al. J Med Chem. 2004 Jul 15;47(15):3892-6. doi: 10.1021/jm031147e. J Med Chem. 2004. PMID: 15239667

7

Imidazole analogues of fluoxetine, a novel class of anti-Candida agents.

Silvestri R, Artico M, La Regina G, Di Pasquali A, De Martino G, D'Auria FD, Nencioni L, Palamara AT. Silvestri R, et al. J Med Chem. 2004 Jul 29;47(16):3924-6. doi: 10.1021/jm049856v. J Med Chem. 2004. PMID: 15267229

8

Arylthioindoles, potent inhibitors of tubulin polymerization.

De Martino G, La Regina G, Coluccia A, Edler MC, Barbera MC, Brancale A, Wilcox E, Hamel E, Artico M, Silvestri R. De Martino G, et al. Among authors: silvestri r. J Med Chem. 2004 Dec 2;47(25):6120-3. doi: 10.1021/jm049360d. J Med Chem. 2004. PMID: 15566282

9

Docking and 3-D QSAR studies on indolyl aryl sulfones. Binding mode exploration at the HIV-1 reverse transcriptase non-nucleoside binding site and design of highly active N-(2-hydroxyethyl)carboxamide and N-(2-hydroxyethyl)carbohydrazide derivatives.

Ragno R, Artico M, De Martino G, La Regina G, Coluccia A, Di Pasquali A, Silvestri R. Ragno R, et al. Among authors: silvestri r. J Med Chem. 2005 Jan 13;48(1):213-23. doi: 10.1021/jm040854k. J Med Chem. 2005. PMID: 15634015

Three-dimensional quantitative structure-activity relationship (3-D QSAR) studies and docking simulations were developed on indolyl aryl sulfones (IASs), a class of novel HIV-1 non-nucleoside reverse transcriptase (RT) inhibitors (Silvestri, et al. J. Med. Chem. 2003, 46, …

Three-dimensional quantitative structure-activity relationship (3-D QSAR) studies and docking simulations were developed on indolyl aryl sul …

10

Comparative study between the polysaccharide-based chiralcel OJ and chiralcel OD CSPSs in chromatographic enantioseparation of imidazole analogues of fluoxetine and miconazole.

Cirilli R, Ferretti R, Gallinella B, La Torre F, La Regina G, Silvestri R. Cirilli R, et al. Among authors: silvestri r. J Sep Sci. 2005 May;28(7):627-34. doi: 10.1002/jssc.200400102. J Sep Sci. 2005. PMID: 15912731

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