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Potentiation of antibiotic activity, and efflux pumps inhibition by (2E)-1-(4-aminophenyl)-3-(4-fluorophenyl)prop-2-en-1-one.
Fundam Clin Pharmacol. 2022 Dec;36(6):1066-1082. doi: 10.1111/fcp.12785. Epub 2022 May 19.
Fundam Clin Pharmacol. 2022.
PMID: 35475507
Antibacterial and antibiotic modifying activity of chalcone (2E)-1-(4'-aminophenyl)-3-(4-methoxyphenyl)-prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps: In vitro and in silico approaches.
Silva J, Esmeraldo Rocha J, da Cunha Xavier J, Sampaio de Freitas T, Douglas Melo Coutinho H, Nogueira Bandeira P, Rodrigues de Oliveira M, Nunes da Rocha M, Machado Marinho E, de Kassio Vieira Monteiro N, Ribeiro LR, Róseo Paula Pessoa Bezerra de Menezes R, Machado Marinho M, Magno Rodrigues Teixeira A, Silva Dos Santos H, Silva Marinho E.
Silva J, et al. Among authors: silva marinho e.
Microb Pathog. 2022 Aug;169:105664. doi: 10.1016/j.micpath.2022.105664. Epub 2022 Jul 5.
Microb Pathog. 2022.
PMID: 35803497
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Synthesis and in silico study of chenodeoxycholic acid and its analogues as an alternative inhibitor of spike glycoprotein of SARS-CoV-2.
Rocha Aguiar G, Leda Gomes de Lemos T, Braz-Filho R, Marques da Fonseca A, Silva Marinho E, Vasconcelos Ribeiro PR, Marques Canuto K, Queiroz Monte FJ.
Rocha Aguiar G, et al. Among authors: silva marinho e.
J Biomol Struct Dyn. 2023 Oct-Nov;41(17):8334-8348. doi: 10.1080/07391102.2022.2133010. Epub 2022 Oct 11.
J Biomol Struct Dyn. 2023.
PMID: 36218138
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Essential Oils from the Genus Piper Promote Antinociception by Modulating TRP Channels and Anti-Inflammatory Effects in Adult Zebrafish.
Pereira WF, Everson da Silva L, do Amaral W, Andrade Rebelo R, Quefi B, Wlisses da Silva A, Silva Marinho E, Borges Leal ALA, Mesquita Cajazeiras FF, Amâncio Ferreira MK, Bezerra Maciel J, Ribeiro Liberato H, Guedes JM, Silva Alencar de Menezes JE, Teixeira AMR, Silva Dos Santosa H.
Pereira WF, et al. Among authors: silva marinho e.
Chem Biodivers. 2024 Mar;21(3):e202301807. doi: 10.1002/cbdv.202301807. Epub 2024 Feb 19.
Chem Biodivers. 2024.
PMID: 38284478
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Trypanocidal potential of synthetic p-aminochalcones: In silico and in vitro evaluation.
Dutra Barroso Gomes N, Paula Magalhães E, Rodrigues Ribeiro L, Cavalcante JW, Morais Gomes Maia M, Cunha da Silva FR, Ali A, Machado Marinho M, Silva Marinho E, Silva Dos Santos H, Costa Martins AM, Róseo Paula Pessoa Bezerra de Menezes R.
Dutra Barroso Gomes N, et al. Among authors: silva marinho e.
Bioorg Chem. 2023 Dec;141:106931. doi: 10.1016/j.bioorg.2023.106931. Epub 2023 Oct 20.
Bioorg Chem. 2023.
PMID: 37879182
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Synthesis, molecular docking, ADMET, and evaluation of the anxiolytic effect in adult zebrafish of synthetic chalcone (E)-3-(4-(dimethylamino)phenyl)-1-(2-hydroxyphenyl)prop-2-en-1-one: An in vivo and in silico approach.
Santos Oliveira L, Kueirislene Amâncio Ferreira M, Wagner de Queiroz Almeida-Neto F, Wlisses da Silva A, Ivo Lima Pinto Filho J, Nunes da Rocha M, Machado Marinho E, Henrique Ferreira Ribeiro W, Machado Marinho M, Silva Marinho E, Eire Silva Alencar de Menezes J, Dos Santos HS.
Santos Oliveira L, et al. Among authors: silva marinho e.
Fundam Clin Pharmacol. 2024 Apr;38(2):290-306. doi: 10.1111/fcp.12960. Epub 2023 Oct 16.
Fundam Clin Pharmacol. 2024.
PMID: 37845792
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