Design, synthesis, and evaluation of metabolism-based analogues of haloperidol incapable of forming MPP+-like species.
Lyles-Eggleston M, Altundas R, Xia J, Sikazwe DM, Fan P, Yang Q, Li S, Zhang W, Zhu X, Schmidt AW, Vanase-Frawley M, Shrihkande A, Villalobos A, Borne RF, Ablordeppey SY.
Lyles-Eggleston M, et al. Among authors: sikazwe dm.
J Med Chem. 2004 Jan 29;47(3):497-508. doi: 10.1021/jm0301033.
J Med Chem. 2004.
PMID: 14736232