Sieńczyk M - Search Results

1

Exploiting the S4-S5 Specificity of Human Neutrophil Proteinase 3 to Improve the Potency of Peptidyl Di(chlorophenyl)-phosphonate Ester Inhibitors: A Kinetic and Molecular Modeling Analysis.

Guarino C, Gruba N, Grzywa R, Dyguda-Kazimierowicz E, Hamon Y, Łȩgowska M, Skoreński M, Dallet-Choisy S, Marchand-Adam S, Kellenberger C, Jenne DE, Sieńczyk M, Lesner A, Gauthier F, Korkmaz B. Guarino C, et al. Among authors: sienczyk m. J Med Chem. 2018 Mar 8;61(5):1858-1870. doi: 10.1021/acs.jmedchem.7b01416. Epub 2018 Feb 26. J Med Chem. 2018. PMID: 29442501

2

Inhibition of trypsin and urokinase by Cbz-amino(4-guanidinophenyl)methanephosphonate aromatic ester derivatives: the influence of the ester group on their biological activity.

Sieńczyk M, Oleksyszyn J. Sieńczyk M, et al. Bioorg Med Chem Lett. 2006 Jun 1;16(11):2886-90. doi: 10.1016/j.bmcl.2006.03.002. Epub 2006 Mar 20. Bioorg Med Chem Lett. 2006. PMID: 16546384

3

The molecular basis of urokinase inhibition: from the nonempirical analysis of intermolecular interactions to the prediction of binding affinity.

Grzywa R, Dyguda-Kazimierowicz E, Sieńczyk M, Feliks M, Sokalski WA, Oleksyszyn J. Grzywa R, et al. Among authors: sienczyk m. J Mol Model. 2007 Jul;13(6-7):677-83. doi: 10.1007/s00894-007-0193-8. Epub 2007 Mar 20. J Mol Model. 2007. PMID: 17587094

4

New potent cathepsin G phosphonate inhibitors.

Sieńczyk M, Lesner A, Wysocka M, Legowska A, Pietrusewicz E, Rolka K, Oleksyszyn J. Sieńczyk M, et al. Bioorg Med Chem. 2008 Oct 1;16(19):8863-7. doi: 10.1016/j.bmc.2008.08.069. Epub 2008 Aug 31. Bioorg Med Chem. 2008. PMID: 18805698

5

Irreversible inhibition of serine proteases - design and in vivo activity of diaryl alpha-aminophosphonate derivatives.

Sieńczyk M, Oleksyszyn J. Sieńczyk M, et al. Curr Med Chem. 2009;16(13):1673-87. doi: 10.2174/092986709788186246. Curr Med Chem. 2009. PMID: 19442139

6

Novel diphenyl esters of peptidyl alpha-aminoalkylphosphonates as inhibitors of chymotrypsin and subtilisin.

Pietrusewicz E, Sieńczyk M, Oleksyszyn J. Pietrusewicz E, et al. Among authors: sienczyk m. J Enzyme Inhib Med Chem. 2009 Dec;24(6):1229-36. doi: 10.3109/14756360902781512. J Enzyme Inhib Med Chem. 2009. PMID: 19912056

7

New aromatic monoesters of alpha-aminoaralkylphosphonic acids as inhibitors of aminopeptidase N/CD13.

Grzywa R, Sokol AM, Sieńczyk M, Radziszewicz M, Kościołek B, Carty MP, Oleksyszyn J. Grzywa R, et al. Among authors: sienczyk m. Bioorg Med Chem. 2010 Apr 15;18(8):2930-6. doi: 10.1016/j.bmc.2010.02.056. Epub 2010 Mar 1. Bioorg Med Chem. 2010. PMID: 20347318

8

Phosphonic pseudopeptides as human neutrophil elastase inhibitors--a combinatorial approach.

Sieńczyk M, Podgórski D, Błażejewska A, Kulbacka J, Saczko J, Oleksyszyn J. Sieńczyk M, et al. Bioorg Med Chem. 2011 Feb 1;19(3):1277-84. doi: 10.1016/j.bmc.2010.12.008. Epub 2010 Dec 9. Bioorg Med Chem. 2011. PMID: 21216608

9

Simple phosphonic inhibitors of human neutrophil elastase.

Sieńczyk M, Winiarski Ł, Kasperkiewicz P, Psurski M, Wietrzyk J, Oleksyszyn J. Sieńczyk M, et al. Bioorg Med Chem Lett. 2011 Mar 1;21(5):1310-4. doi: 10.1016/j.bmcl.2011.01.083. Epub 2011 Jan 22. Bioorg Med Chem Lett. 2011. PMID: 21315589

10

Surface plasmon resonance imaging biosensor for cathepsin G based on a potent inhibitor: development and applications.

Gorodkiewicz E, Sieńczyk M, Regulska E, Grzywa R, Pietrusewicz E, Lesner A, Lukaszewski Z. Gorodkiewicz E, et al. Among authors: sienczyk m. Anal Biochem. 2012 Apr 15;423(2):218-23. doi: 10.1016/j.ab.2012.01.033. Epub 2012 Feb 7. Anal Biochem. 2012. PMID: 22369897

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