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Hit-to-Lead Optimization of Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists with a Diphenylmethane-Scaffold: Design, Synthesis, and Biological Study.
Chiellini G, Nesi G, Sestito S, Chiarugi S, Runfola M, Espinoza S, Sabatini M, Bellusci L, Laurino A, Cichero E, Gainetdinov RR, Fossa P, Raimondi L, Zucchi R, Rapposelli S. Chiellini G, et al. Among authors: sestito s. J Med Chem. 2016 Nov 10;59(21):9825-9836. doi: 10.1021/acs.jmedchem.6b01092. Epub 2016 Oct 21. J Med Chem. 2016. PMID: 27731647
New Insights into the Potential Roles of 3-Iodothyronamine (T1AM) and Newly Developed Thyronamine-Like TAAR1 Agonists in Neuroprotection.
Bellusci L, Laurino A, Sabatini M, Sestito S, Lenzi P, Raimondi L, Rapposelli S, Biagioni F, Fornai F, Salvetti A, Rossi L, Zucchi R, Chiellini G. Bellusci L, et al. Among authors: sestito s. Front Pharmacol. 2017 Dec 12;8:905. doi: 10.3389/fphar.2017.00905. eCollection 2017. Front Pharmacol. 2017. PMID: 29311919 Free PMC article.
Memantine prodrug as a new agent for Alzheimer's Disease.
Sestito S, Daniele S, Pietrobono D, Citi V, Bellusci L, Chiellini G, Calderone V, Martini C, Rapposelli S. Sestito S, et al. Sci Rep. 2019 Mar 15;9(1):4612. doi: 10.1038/s41598-019-40925-8. Sci Rep. 2019. PMID: 30874573 Free PMC article.
A patent update on PDK1 inhibitors (2015-present).
Sestito S, Rapposelli S. Sestito S, et al. Expert Opin Ther Pat. 2019 Apr;29(4):271-282. doi: 10.1080/13543776.2019.1597852. Epub 2019 Mar 29. Expert Opin Ther Pat. 2019. PMID: 30897008 Review.
Collecting data through high throughput in vitro early toxicity and off-target liability assays to rapidly identify limitations of novel thyromimetics.
Runfola M, Sestito S, Gul S, Chiellini G, Rapposelli S. Runfola M, et al. Among authors: sestito s. Data Brief. 2020 Jan 31;29:105206. doi: 10.1016/j.dib.2020.105206. eCollection 2020 Apr. Data Brief. 2020. PMID: 32071982 Free PMC article.
The data reported herein support our research article entitled "Design, synthesis and biological evaluation of novel TRbeta selective agonists sustained by ADME-Toxicity analysis" by Runfola M., Sestito S., et al. [1]....
The data reported herein support our research article entitled "Design, synthesis and biological evaluation of novel TRbeta selective agonis …
105 results