Schmidt B - Search Results

1

Proteasome inhibition potentiates Kv1.3 potassium channel expression as therapeutic target in drug-sensitive and -resistant human melanoma cells.

Cammann C, Kulla J, Wiebusch L, Walz C, Zhao F, Lowinus T, Topfstedt E, Mishra N, Henklein P, Bommhardt U, Bossaller L, Hagemeier C, Schadendorf D, Schmidt B, Paschen A, Seifert U. Cammann C, et al. Among authors: schmidt b. Biomed Pharmacother. 2023 Dec;168:115635. doi: 10.1016/j.biopha.2023.115635. Epub 2023 Oct 8. Biomed Pharmacother. 2023. PMID: 37816303 Free article.

2

Combined effect of proteasome and calpain inhibition on cisplatin-resistant human melanoma cells.

Młynarczuk-Biały I, Roeckmann H, Kuckelkorn U, Schmidt B, Umbreen S, Gołab J, Ludwig A, Montag C, Wiebusch L, Hagemeier C, Schadendorf D, Kloetzel PM, Seifert U. Młynarczuk-Biały I, et al. Among authors: schmidt b. Cancer Res. 2006 Aug 1;66(15):7598-605. doi: 10.1158/0008-5472.CAN-05-2614. Cancer Res. 2006. PMID: 16885359

3

Biodistribution and Efficacy Studies of the Proteasome Inhibitor BSc2118 in a Mouse Melanoma Model.

Mlynarczuk-Bialy I, Doeppner TR, Golab J, Nowis D, Wilczynski GM, Parobczak K, Wigand ME, Hajdamowicz M, Biały LP, Aniolek O, Henklein P, Bähr M, Schmidt B, Kuckelkorn U, Kloetzel PM. Mlynarczuk-Bialy I, et al. Among authors: schmidt b. Transl Oncol. 2014 Oct 24;7(5):570-9. doi: 10.1016/j.tranon.2014.07.002. eCollection 2014 Oct. Transl Oncol. 2014. PMID: 25389452 Free PMC article.

4

α-Keto phenylamides as P1'-extended proteasome inhibitors.

Voss C, Scholz C, Knorr S, Beck P, Stein ML, Zall A, Kuckelkorn U, Kloetzel PM, Groll M, Hamacher K, Schmidt B. Voss C, et al. Among authors: schmidt b. ChemMedChem. 2014 Nov;9(11):2557-64. doi: 10.1002/cmdc.201402244. Epub 2014 Aug 1. ChemMedChem. 2014. PMID: 25087721

5

Tripeptide mimetics inhibit the 20 S proteasome by covalent bonding to the active threonines.

Braun HA, Umbreen S, Groll M, Kuckelkorn U, Mlynarczuk I, Wigand ME, Drung I, Kloetzel PM, Schmidt B. Braun HA, et al. Among authors: schmidt b. J Biol Chem. 2005 Aug 5;280(31):28394-401. doi: 10.1074/jbc.M502453200. Epub 2005 May 26. J Biol Chem. 2005. PMID: 15919666 Free article.

6

Elastase-like Activity Is Dominant to Chymotrypsin-like Activity in 20S Proteasome's β5 Catalytic Subunit.

Bensinger D, Neumann T, Scholz C, Voss C, Knorr S, Kuckelkorn U, Hamacher K, Kloetzel PM, Schmidt B. Bensinger D, et al. Among authors: schmidt b. ACS Chem Biol. 2016 Jul 15;11(7):1800-4. doi: 10.1021/acschembio.6b00023. Epub 2016 May 2. ACS Chem Biol. 2016. PMID: 27111844

7

Cell-Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit.

Stubba D, Bensinger D, Steinbacher J, Proskurjakov L, Salcedo Gómez Á, Schmidt U, Roth S, Schmitz K, Schmidt B. Stubba D, et al. Among authors: schmidt b, schmidt u. ChemMedChem. 2019 Dec 4;14(23):2005-2022. doi: 10.1002/cmdc.201900472. Epub 2019 Nov 12. ChemMedChem. 2019. PMID: 31675179 Free PMC article.

8

Inhibition of gamma-secretase by the CK1 inhibitor IC261 does not depend on CK1delta.

Höttecke N, Liebeck M, Baumann K, Schubenel R, Winkler E, Steiner H, Schmidt B. Höttecke N, et al. Among authors: schmidt b. Bioorg Med Chem Lett. 2010 May 1;20(9):2958-63. doi: 10.1016/j.bmcl.2010.02.110. Epub 2010 Mar 4. Bioorg Med Chem Lett. 2010. PMID: 20350806

9

Modification of a promiscuous inhibitor shifts the inhibition from γ-secretase to FLT-3.

Amombo GM, Kramer T, Lo Monte F, Göring S, Fach M, Smith S, Kolb S, Schubenel R, Baumann K, Schmidt B. Amombo GM, et al. Among authors: schmidt b. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7634-40. doi: 10.1016/j.bmcl.2012.10.016. Epub 2012 Oct 11. Bioorg Med Chem Lett. 2012. PMID: 23107479

10

Virtual Screening Identifies Irreversible FMS-like Tyrosine Kinase 3 Inhibitors with Activity toward Resistance-Conferring Mutations.

Bensinger D, Stubba D, Cremer A, Kohl V, Waßmer T, Stuckert J, Engemann V, Stegmaier K, Schmitz K, Schmidt B. Bensinger D, et al. Among authors: schmidt b. J Med Chem. 2019 Mar 14;62(5):2428-2446. doi: 10.1021/acs.jmedchem.8b01714. Epub 2019 Feb 25. J Med Chem. 2019. PMID: 30742435

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

4,120 results

Search Page