Schirmeister T - Search Results

1

Bistacrines as potential antitrypanosomal agents.

Schmidt I, Göllner S, Fuß A, Stich A, Kucharski A, Schirmeister T, Katzowitsch E, Bruhn H, Miliu A, Krauth-Siegel RL, Holzgrabe U. Schmidt I, et al. Among authors: schirmeister t. Bioorg Med Chem. 2017 Aug 15;25(16):4526-4531. doi: 10.1016/j.bmc.2017.06.051. Epub 2017 Jul 1. Bioorg Med Chem. 2017. PMID: 28698054

2

Development and validation of a separation method for the diastereomers and enantiomers of aziridine-type protease inhibitors.

Bitar Y, Degel B, Schirmeister T, Holzgrabe U. Bitar Y, et al. Among authors: schirmeister t. Electrophoresis. 2005 Jun;26(12):2313-9. doi: 10.1002/elps.200410302. Electrophoresis. 2005. PMID: 15912540

3

Comparison of the separation of aziridine isomers applying heptakis(2,3-di-O-methyl-6-sulfato)beta-CD and heptakis(2,3-di-O-acetyl-6-sulfato)beta-CD in aqueous and nonaqueous systems.

Bitar Y, Degel B, Schirmeister T, Holzgrabe U. Bitar Y, et al. Among authors: schirmeister t. Electrophoresis. 2005 Oct;26(20):3897-903. doi: 10.1002/elps.200500176. Electrophoresis. 2005. PMID: 16167307

4

Screening of electrophilic compounds yields an aziridinyl peptide as new active-site directed SARS-CoV main protease inhibitor.

Martina E, Stiefl N, Degel B, Schulz F, Breuning A, Schiller M, Vicik R, Baumann K, Ziebuhr J, Schirmeister T. Martina E, et al. Among authors: schirmeister t. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5365-9. doi: 10.1016/j.bmcl.2005.09.012. Epub 2005 Oct 10. Bioorg Med Chem Lett. 2005. PMID: 16216498 Free PMC article.

5

A new lead for nonpeptidic active-site-directed inhibitors of the severe acute respiratory syndrome coronavirus main protease discovered by a combination of screening and docking methods.

Kaeppler U, Stiefl N, Schiller M, Vicik R, Breuning A, Schmitz W, Rupprecht D, Schmuck C, Baumann K, Ziebuhr J, Schirmeister T. Kaeppler U, et al. Among authors: schirmeister t. J Med Chem. 2005 Nov 3;48(22):6832-42. doi: 10.1021/jm0501782. J Med Chem. 2005. PMID: 16250642

6

Aziridine-2,3-dicarboxylate inhibitors targeting the major cysteine protease of Trypanosoma brucei as lead trypanocidal agents.

Vicik R, Hoerr V, Glaser M, Schultheis M, Hansell E, McKerrow JH, Holzgrabe U, Caffrey CR, Ponte-Sucre A, Moll H, Stich A, Schirmeister T. Vicik R, et al. Among authors: schirmeister t. Bioorg Med Chem Lett. 2006 May 15;16(10):2753-7. doi: 10.1016/j.bmcl.2006.02.026. Epub 2006 Mar 3. Bioorg Med Chem Lett. 2006. PMID: 16516467

7

Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors.

Micale N, Ettari R, Schirmeister T, Evers A, Gelhaus C, Leippe M, Zappalà M, Grasso S. Micale N, et al. Among authors: schirmeister t. Bioorg Med Chem. 2009 Sep 15;17(18):6505-11. doi: 10.1016/j.bmc.2009.08.013. Epub 2009 Aug 12. Bioorg Med Chem. 2009. PMID: 19709887

8

Michael acceptor based antiplasmodial and antitrypanosomal cysteine protease inhibitors with unusual amino acids.

Breuning A, Degel B, Schulz F, Büchold C, Stempka M, Machon U, Heppner S, Gelhaus C, Leippe M, Leyh M, Kisker C, Rath J, Stich A, Gut J, Rosenthal PJ, Schmuck C, Schirmeister T. Breuning A, et al. Among authors: schirmeister t. J Med Chem. 2010 Mar 11;53(5):1951-63. doi: 10.1021/jm900946n. J Med Chem. 2010. PMID: 20131843

9

Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors.

Bova F, Ettari R, Micale N, Carnovale C, Schirmeister T, Gelhaus C, Leippe M, Grasso S, Zappalà M. Bova F, et al. Among authors: schirmeister t. Bioorg Med Chem. 2010 Jul 15;18(14):4928-38. doi: 10.1016/j.bmc.2010.06.010. Epub 2010 Jun 10. Bioorg Med Chem. 2010. PMID: 20598553

10

Allicin and derivates are cysteine protease inhibitors with antiparasitic activity.

Waag T, Gelhaus C, Rath J, Stich A, Leippe M, Schirmeister T. Waag T, et al. Among authors: schirmeister t. Bioorg Med Chem Lett. 2010 Sep 15;20(18):5541-3. doi: 10.1016/j.bmcl.2010.07.062. Epub 2010 Aug 6. Bioorg Med Chem Lett. 2010. PMID: 20692829

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