Schütz J - Search Results

1

Functionalization of the carbonyl group in position 6 of morphinan-6-ones. Development of novel 6-amino and 6-guanidino substituted 14-alkoxymorphinans.

Schmidhammer H, Spetea M, Windisch P, Schütz J, Riba P, Al-Khrasani M, Furst S. Schmidhammer H, et al. Among authors: schutz j. Curr Pharm Des. 2013;19(42):7391-9. doi: 10.2174/138161281942140105164804. Curr Pharm Des. 2013. PMID: 23448473 Review.

2

Synthesis and biological evaluation of 14-alkoxymorphinans. 17. Highly delta opioid receptor selective 14-alkoxy-substituted indolo- and benzofuromorphinans.

Schütz J, Dersch CM, Horel R, Spetea M, Koch M, Meditz R, Greiner E, Rothman RB, Schmidhammer H. Schütz J, et al. J Med Chem. 2002 Nov 21;45(24):5378-83. doi: 10.1021/jm020940p. J Med Chem. 2002. PMID: 12431065

3

Synthesis and pharmacological activities of 6-glycine substituted 14-phenylpropoxymorphinans, a novel class of opioids with high opioid receptor affinities and antinociceptive potencies.

Spetea M, Windisch P, Guo Y, Bileviciute-Ljungar I, Schütz J, Asim MF, Berzetei-Gurske IP, Riba P, Kiraly K, Fürst S, Al-Khrasani M, Schmidhammer H. Spetea M, et al. Among authors: schutz j. J Med Chem. 2011 Feb 24;54(4):980-8. doi: 10.1021/jm101211p. Epub 2011 Jan 14. J Med Chem. 2011. PMID: 21235243 Free PMC article.

4

Synthesis and biological evaluation of 14-alkoxymorphinans. 20. 14-phenylpropoxymetopon: an extremely powerful analgesic.

Schütz J, Spetea M, Koch M, Aceto MD, Harris LS, Coop A, Schmidhammer H. Schütz J, et al. J Med Chem. 2003 Sep 11;46(19):4182-7. doi: 10.1021/jm030878b. J Med Chem. 2003. PMID: 12954070

5

In vitro opioid activity profiles of 6-amino acid substituted derivatives of 14-O-methyloxymorphone.

Spetea M, Friedmann T, Riba P, Schütz J, Wunder G, Langer T, Schmidhammer H, Fürst S. Spetea M, et al. Among authors: schutz j. Eur J Pharmacol. 2004 Jan 12;483(2-3):301-8. doi: 10.1016/j.ejphar.2003.10.049. Eur J Pharmacol. 2004. PMID: 14729121

6

Mechanistic diversity of the van Leusen reaction applied to 6-ketomorphinans and synthetic potential of the resulting acrylonitrile substructures.

Schütz J, Windisch P, Kristeva E, Wurst K, Ongania KH, Horvath UE, Schottenberger H, Laus G, Schmidhammer H. Schütz J, et al. J Org Chem. 2005 Jun 24;70(13):5323-6. doi: 10.1021/jo050362v. J Org Chem. 2005. PMID: 15960541

7

Morphinans and isoquinolines: acetylcholinesterase inhibition, pharmacophore modeling, and interaction with opioid receptors.

Schuster D, Spetea M, Music M, Rief S, Fink M, Kirchmair J, Schütz J, Wolber G, Langer T, Stuppner H, Schmidhammer H, Rollinger JM. Schuster D, et al. Among authors: schutz j. Bioorg Med Chem. 2010 Jul 15;18(14):5071-80. doi: 10.1016/j.bmc.2010.05.071. Epub 2010 Jun 2. Bioorg Med Chem. 2010. PMID: 20580236

8

Binding characteristics of [3H]14-methoxymetopon, a high affinity mu-opioid receptor agonist.

Spetea M, Tóth F, Schütz J, Otvös F, Tóth G, Benyhe S, Borsodi A, Schmidhammer H. Spetea M, et al. Among authors: schutz j. Eur J Neurosci. 2003 Jul;18(2):290-5. doi: 10.1046/j.1460-9568.2003.02744.x. Eur J Neurosci. 2003. PMID: 12887410

9

Peripherally mediated antinociception of the mu-opioid receptor agonist 2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid (HS-731) after subcutaneous and oral administration in rats with carrageenan-induced hindpaw inflammation.

Bileviciute-Ljungar I, Spetea M, Guo Y, Schütz J, Windisch P, Schmidhammer H. Bileviciute-Ljungar I, et al. Among authors: schutz j. J Pharmacol Exp Ther. 2006 Apr;317(1):220-7. doi: 10.1124/jpet.105.096032. Epub 2005 Dec 8. J Pharmacol Exp Ther. 2006. PMID: 16339394

10

Peripheral versus central antinociceptive actions of 6-amino acid-substituted derivatives of 14-O-methyloxymorphone in acute and inflammatory pain in the rat.

Fürst S, Riba P, Friedmann T, Tímar J, Al-Khrasani M, Obara I, Makuch W, Spetea M, Schütz J, Przewlocki R, Przewlocka B, Schmidhammer H. Fürst S, et al. Among authors: schutz j. J Pharmacol Exp Ther. 2005 Feb;312(2):609-18. doi: 10.1124/jpet.104.075176. Epub 2004 Sep 21. J Pharmacol Exp Ther. 2005. PMID: 15383636

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