Scalvini L - Search Results

1

Fighting tertiary mutations in EGFR-driven lung-cancers: Current advances and future perspectives in medicinal chemistry.

Scalvini L, Castelli R, La Monica S, Tiseo M, Alfieri R. Scalvini L, et al. Biochem Pharmacol. 2021 Aug;190:114643. doi: 10.1016/j.bcp.2021.114643. Epub 2021 Jun 10. Biochem Pharmacol. 2021. PMID: 34097913 Review.

2

Amino Acid Derivatives as Palmitoylethanolamide Prodrugs: Synthesis, In Vitro Metabolism and In Vivo Plasma Profile in Rats.

Vacondio F, Bassi M, Silva C, Castelli R, Carmi C, Scalvini L, Lodola A, Vivo V, Flammini L, Barocelli E, Mor M, Rivara S. Vacondio F, et al. Among authors: scalvini l. PLoS One. 2015 Jun 8;10(6):e0128699. doi: 10.1371/journal.pone.0128699. eCollection 2015. PLoS One. 2015. PMID: 26053855 Free PMC article.

3

Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines.

Castelli R, Scalvini L, Vacondio F, Lodola A, Anselmi M, Vezzosi S, Carmi C, Bassi M, Ferlenghi F, Rivara S, Møller IR, Rand KD, Daglian J, Wei D, Dotsey EY, Ahmed F, Jung KM, Stella N, Singh S, Mor M, Piomelli D. Castelli R, et al. Among authors: scalvini l. J Med Chem. 2020 Feb 13;63(3):1261-1280. doi: 10.1021/acs.jmedchem.9b01679. Epub 2019 Dec 2. J Med Chem. 2020. PMID: 31714779

4

Drug-gut microbiota metabolic interactions: the case of UniPR1331, selective antagonist of the Eph-ephrin system, in mice.

Ferlenghi F, Castelli R, Scalvini L, Giorgio C, Corrado M, Tognolini M, Mor M, Lodola A, Vacondio F. Ferlenghi F, et al. Among authors: scalvini l. J Pharm Biomed Anal. 2020 Feb 20;180:113067. doi: 10.1016/j.jpba.2019.113067. Epub 2019 Dec 23. J Pharm Biomed Anal. 2020. PMID: 31891876

5

Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties.

Incerti M, Russo S, Corrado M, Giorgio C, Ballabeni V, Chiodelli P, Rusnati M, Scalvini L, Callegari D, Castelli R, Vacondio F, Ferlenghi F, Tognolini M, Lodola A. Incerti M, et al. Among authors: scalvini l. Eur J Med Chem. 2020 Mar 1;189:112083. doi: 10.1016/j.ejmech.2020.112083. Epub 2020 Jan 22. Eur J Med Chem. 2020. PMID: 32000051

6

A sulfonyl fluoride derivative inhibits EGFR^{L858R/T790M/C797S} by covalent modification of the catalytic lysine.

Ferlenghi F, Scalvini L, Vacondio F, Castelli R, Bozza N, Marseglia G, Rivara S, Lodola A, La Monica S, Minari R, Petronini PG, Alfieri R, Tiseo M, Mor M. Ferlenghi F, et al. Among authors: scalvini l. Eur J Med Chem. 2021 Dec 5;225:113786. doi: 10.1016/j.ejmech.2021.113786. Epub 2021 Aug 27. Eur J Med Chem. 2021. PMID: 34464874

7

Protein-Protein Interaction Inhibitors Targeting the Eph-Ephrin System with a Focus on Amino Acid Conjugates of Bile Acids.

Guidetti L, Castelli R, Scalvini L, Ferlenghi F, Corrado M, Giorgio C, Tognolini M, Lodola A. Guidetti L, et al. Among authors: scalvini l. Pharmaceuticals (Basel). 2022 Jan 24;15(2):137. doi: 10.3390/ph15020137. Pharmaceuticals (Basel). 2022. PMID: 35215250 Free PMC article. Review.

8

Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity.

Guidetti L, Zappia A, Scalvini L, Ferrari FR, Giorgio C, Castelli R, Galvani F, Vacondio F, Rivara S, Mor M, Urbinati C, Rusnati M, Tognolini M, Lodola A. Guidetti L, et al. Among authors: scalvini l. J Chem Inf Model. 2023 Nov 13;63(21):6900-6911. doi: 10.1021/acs.jcim.3c01064. Epub 2023 Nov 1. J Chem Inf Model. 2023. PMID: 37910792 Free PMC article.

9

Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations.

Lodola A, Callegari D, Scalvini L, Rivara S, Mor M. Lodola A, et al. Among authors: scalvini l. Methods Mol Biol. 2020;2114:307-337. doi: 10.1007/978-1-0716-0282-9_19. Methods Mol Biol. 2020. PMID: 32016901 Review.

10

Pharmacological characterization of second generation FXR agonists as effective EphA2 antagonists: A successful application of target hopping approach.

Ferrari FR, Giorgio C, Zappia A, Ballabeni V, Bertoni S, Barocelli E, Scalvini L, Galvani F, Mor M, Lodola A, Tognolini M. Ferrari FR, et al. Among authors: scalvini l. Biochem Pharmacol. 2023 Mar;209:115452. doi: 10.1016/j.bcp.2023.115452. Epub 2023 Feb 13. Biochem Pharmacol. 2023. PMID: 36792038

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