Sbardella G - Search Results

1

Arginine Demethylation of G3BP1 Promotes Stress Granule Assembly.

Tsai WC, Gayatri S, Reineke LC, Sbardella G, Bedford MT, Lloyd RE. Tsai WC, et al. Among authors: sbardella g. J Biol Chem. 2016 Oct 21;291(43):22671-22685. doi: 10.1074/jbc.M116.739573. Epub 2016 Sep 6. J Biol Chem. 2016. PMID: 27601476 Free PMC article.

2

NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors.

Cipriano A, Viviano M, Feoli A, Milite C, Sarno G, Castellano S, Sbardella G. Cipriano A, et al. Among authors: sbardella g. J Med Chem. 2023 Sep 14;66(17):11632-11655. doi: 10.1021/acs.jmedchem.3c00770. Epub 2023 Aug 31. J Med Chem. 2023. PMID: 37650225 Free PMC article. Review.

3

Synthesis and biological validation of novel synthetic histone/protein methyltransferase inhibitors.

Mai A, Valente S, Cheng D, Perrone A, Ragno R, Simeoni S, Sbardella G, Brosch G, Nebbioso A, Conte M, Altucci L, Bedford MT. Mai A, et al. Among authors: sbardella g. ChemMedChem. 2007 Jul;2(7):987-91. doi: 10.1002/cmdc.200700023. ChemMedChem. 2007. PMID: 17458842 No abstract available.

4

epigenetic multiple ligands: mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors.

Mai A, Cheng D, Bedford MT, Valente S, Nebbioso A, Perrone A, Brosch G, Sbardella G, De Bellis F, Miceli M, Altucci L. Mai A, et al. Among authors: sbardella g. J Med Chem. 2008 Apr 10;51(7):2279-90. doi: 10.1021/jm701595q. Epub 2008 Mar 19. J Med Chem. 2008. PMID: 18348515

5

Design, synthesis and biological evaluation of carboxy analogues of arginine methyltransferase inhibitor 1 (AMI-1).

Castellano S, Milite C, Ragno R, Simeoni S, Mai A, Limongelli V, Novellino E, Bauer I, Brosch G, Spannhoff A, Cheng D, Bedford MT, Sbardella G. Castellano S, et al. Among authors: sbardella g. ChemMedChem. 2010 Mar 1;5(3):398-414. doi: 10.1002/cmdc.200900459. ChemMedChem. 2010. PMID: 20091730

6

Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees.

Spannhoff A, Kim YK, Raynal NJ, Gharibyan V, Su MB, Zhou YY, Li J, Castellano S, Sbardella G, Issa JP, Bedford MT. Spannhoff A, et al. Among authors: sbardella g. EMBO Rep. 2011 Mar;12(3):238-43. doi: 10.1038/embor.2011.9. Epub 2011 Feb 18. EMBO Rep. 2011. PMID: 21331099 Free PMC article.

7

Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.

Cheng D, Valente S, Castellano S, Sbardella G, Di Santo R, Costi R, Bedford MT, Mai A. Cheng D, et al. Among authors: sbardella g. J Med Chem. 2011 Jul 14;54(13):4928-32. doi: 10.1021/jm200453n. Epub 2011 Jun 13. J Med Chem. 2011. PMID: 21612300 Free PMC article.

8

Identification of small-molecule enhancers of arginine methylation catalyzed by coactivator-associated arginine methyltransferase 1.

Castellano S, Spannhoff A, Milite C, Dal Piaz F, Cheng D, Tosco A, Viviano M, Yamani A, Cianciulli A, Sala M, Cura V, Cavarelli J, Novellino E, Mai A, Bedford MT, Sbardella G. Castellano S, et al. Among authors: sbardella g. J Med Chem. 2012 Nov 26;55(22):9875-90. doi: 10.1021/jm301097p. Epub 2012 Nov 2. J Med Chem. 2012. PMID: 23095008 Free PMC article.

9

A TR-FRET-based functional assay for screening activators of CARM1.

Zeng H, Wu J, Bedford MT, Sbardella G, Hoffmann FM, Bi K, Xu W. Zeng H, et al. Among authors: sbardella g. Chembiochem. 2013 May 10;14(7):827-35. doi: 10.1002/cbic.201300029. Epub 2013 Apr 12. Chembiochem. 2013. PMID: 23585185 Free PMC article.

10

Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1.

van Haren MJ, Marechal N, Troffer-Charlier N, Cianciulli A, Sbardella G, Cavarelli J, Martin NI. van Haren MJ, et al. Among authors: sbardella g. Proc Natl Acad Sci U S A. 2017 Apr 4;114(14):3625-3630. doi: 10.1073/pnas.1618401114. Epub 2017 Mar 22. Proc Natl Acad Sci U S A. 2017. PMID: 28330993 Free PMC article.

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