Sawada GA - Search Results

1

QSAR Model of Unbound Brain-to-Plasma Partition Coefficient, K_p,uu,brain: Incorporating P-glycoprotein Efflux as a Variable.

Dolgikh E, Watson IA, Desai PV, Sawada GA, Morton S, Jones TM, Raub TJ. Dolgikh E, et al. Among authors: sawada ga. J Chem Inf Model. 2016 Nov 28;56(11):2225-2233. doi: 10.1021/acs.jcim.6b00229. Epub 2016 Oct 13. J Chem Inf Model. 2016. PMID: 27684523

2

Integration of in silico and in vitro tools for scaffold optimization during drug discovery: predicting P-glycoprotein efflux.

Desai PV, Sawada GA, Watson IA, Raub TJ. Desai PV, et al. Among authors: sawada ga. Mol Pharm. 2013 Apr 1;10(4):1249-61. doi: 10.1021/mp300555n. Epub 2013 Mar 1. Mol Pharm. 2013. PMID: 23363443

3

Chalcogenopyrylium dyes as inhibitors/modulators of P-glycoprotein in multidrug-resistant cells.

Sawada GA, Raub TJ, William Higgins J, Brennan NK, Moore TM, Tombline G, Detty MR. Sawada GA, et al. Bioorg Med Chem. 2008 Nov 15;16(22):9745-56. doi: 10.1016/j.bmc.2008.09.065. Epub 2008 Sep 30. Bioorg Med Chem. 2008. PMID: 18849167

4

Breast cancer resistance protein interacts with various compounds in vitro, but plays a minor role in substrate efflux at the blood-brain barrier.

Zhao R, Raub TJ, Sawada GA, Kasper SC, Bacon JA, Bridges AS, Pollack GM. Zhao R, et al. Among authors: sawada ga. Drug Metab Dispos. 2009 Jun;37(6):1251-8. doi: 10.1124/dmd.108.025064. Epub 2009 Mar 9. Drug Metab Dispos. 2009. PMID: 19273529 Free PMC article.

5

Brain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma Xenograft.

Raub TJ, Wishart GN, Kulanthaivel P, Staton BA, Ajamie RT, Sawada GA, Gelbert LM, Shannon HE, Sanchez-Martinez C, De Dios A. Raub TJ, et al. Among authors: sawada ga. Drug Metab Dispos. 2015 Sep;43(9):1360-71. doi: 10.1124/dmd.114.062745. Epub 2015 Jul 6. Drug Metab Dispos. 2015. PMID: 26149830

6

In Silico and in Vitro Assessment of OATP1B1 Inhibition in Drug Discovery.

Danielson ML, Sawada GA, Raub TJ, Desai PV. Danielson ML, et al. Among authors: sawada ga. Mol Pharm. 2018 Aug 6;15(8):3060-3068. doi: 10.1021/acs.molpharmaceut.8b00168. Epub 2018 Jul 5. Mol Pharm. 2018. PMID: 29927611

7

Expression of a widely distributed, novel sulfated membrane glycoprotein by bovine endothelia and certain transporting epithelia.

Raub TJ, Sawada GA, Kuentzel SL. Raub TJ, et al. Among authors: sawada ga. J Histochem Cytochem. 1994 Sep;42(9):1237-50. doi: 10.1177/42.9.8064131. J Histochem Cytochem. 1994. PMID: 8064131

8

ATP occlusion by P-glycoprotein as a surrogate measure for drug coupling.

Tombline G, Holt JJ, Gannon MK, Donnelly DJ, Wetzel B, Sawada GA, Raub TJ, Detty MR. Tombline G, et al. Among authors: sawada ga. Biochemistry. 2008 Mar 11;47(10):3294-307. doi: 10.1021/bi7021393. Epub 2008 Feb 15. Biochemistry. 2008. PMID: 18275155

9

Permeability of bovine brain microvessel endothelial cells in vitro: barrier tightening by a factor released from astroglioma cells.

Raub TJ, Kuentzel SL, Sawada GA. Raub TJ, et al. Among authors: sawada ga. Exp Cell Res. 1992 Apr;199(2):330-40. doi: 10.1016/0014-4827(92)90442-b. Exp Cell Res. 1992. PMID: 1347502

10

Transcellular permeability of chlorpromazine demonstrating the roles of protein binding and membrane partitioning.

Sawada GA, Ho NF, Williams LR, Barsuhn CL, Raub TJ. Sawada GA, et al. Pharm Res. 1994 May;11(5):665-73. doi: 10.1023/a:1018916027099. Pharm Res. 1994. PMID: 8058634

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