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Structural and Activity Relationships of 6-Sulfonyl-8-Nitrobenzothiazinones as Antitubercular Agents.
J Med Chem. 2021 Oct 14;64(19):14526-14539. doi: 10.1021/acs.jmedchem.1c01049. Epub 2021 Oct 5.
J Med Chem. 2021.
PMID: 34609861
Development of 3,5-Dinitrophenyl-Containing 1,2,4-Triazoles and Their Trifluoromethyl Analogues as Highly Efficient Antitubercular Agents Inhibiting Decaprenylphosphoryl-β-d-ribofuranose 2'-Oxidase.
Karabanovich G, Dušek J, Savková K, Pavliš O, Pávková I, Korábečný J, Kučera T, Kočová Vlčková H, Huszár S, Konyariková Z, Konečná K, Jand'ourek O, Stolaříková J, Korduláková J, Vávrová K, Pávek P, Klimešová V, Hrabálek A, Mikušová K, Roh J.
Karabanovich G, et al. Among authors: savkova k.
J Med Chem. 2019 Sep 12;62(17):8115-8139. doi: 10.1021/acs.jmedchem.9b00912. Epub 2019 Aug 22.
J Med Chem. 2019.
PMID: 31393122
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Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents.
Liu L, Kong C, Fumagalli M, Savková K, Xu Y, Huszár S, Sammartino JC, Fan D, Chiarelli LR, Mikušová K, Sun Z, Qiao C.
Liu L, et al. Among authors: savkova k.
Eur J Med Chem. 2020 Dec 15;208:112773. doi: 10.1016/j.ejmech.2020.112773. Epub 2020 Aug 30.
Eur J Med Chem. 2020.
PMID: 32898793
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Hydride-induced Meisenheimer complex formation reflects activity of nitro aromatic anti-tuberculosis compounds.
Liu R, Markley L, Miller PA, Franzblau S, Shetye G, Ma R, Savková K, Mikušová K, Lee BS, Pethe K, Moraski GC, Miller MJ.
Liu R, et al. Among authors: savkova k.
RSC Med Chem. 2021 Jan 4;12(1):62-72. doi: 10.1039/d0md00390e. eCollection 2021 Jan 1.
RSC Med Chem. 2021.
PMID: 34046598
Free PMC article.
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Biosynthesis of Galactan in Mycobacterium tuberculosis as a Viable TB Drug Target?
Konyariková Z, Savková K, Kozmon S, Mikušová K.
Konyariková Z, et al. Among authors: savkova k.
Antibiotics (Basel). 2020 Jan 6;9(1):20. doi: 10.3390/antibiotics9010020.
Antibiotics (Basel). 2020.
PMID: 31935842
Free PMC article.
Review.
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An ABC transporter Wzm-Wzt catalyzes translocation of lipid-linked galactan across the plasma membrane in mycobacteria.
Savková K, Huszár S, Baráth P, Pakanová Z, Kozmon S, Vancová M, Tesařová M, Blaško J, Kaliňák M, Singh V, Korduláková J, Mikušová K.
Savková K, et al.
Proc Natl Acad Sci U S A. 2021 Apr 27;118(17):e2023663118. doi: 10.1073/pnas.2023663118.
Proc Natl Acad Sci U S A. 2021.
PMID: 33879617
Free PMC article.
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Compartmentalization of galactan biosynthesis in mycobacteria.
Savková K, Danchenko M, Fabianová V, Bellová J, Bencúrová M, Huszár S, Korduláková J, Siváková B, Baráth P, Mikušová K.
Savková K, et al.
J Biol Chem. 2024 Mar;300(3):105768. doi: 10.1016/j.jbc.2024.105768. Epub 2024 Feb 16.
J Biol Chem. 2024.
PMID: 38367664
Free PMC article.
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Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity.
Fan D, Wang B, Stelitano G, Savková K, Riabova O, Shi R, Wu X, Chiarelli LR, Mikušová K, Makarov V, Lu Y, Hong Y, Qiao C.
Fan D, et al. Among authors: savkova k.
Biomedicines. 2023 Jul 12;11(7):1975. doi: 10.3390/biomedicines11071975.
Biomedicines. 2023.
PMID: 37509615
Free PMC article.
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