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Discovery of Potent Indolyl-Hydrazones as Kinase Inhibitors for Breast Cancer: Synthesis, X-ray Single-Crystal Analysis, and In Vitro and In Vivo Anti-Cancer Activity Evaluation.
Pharmaceuticals (Basel). 2023 Dec 13;16(12):1724. doi: 10.3390/ph16121724.
Pharmaceuticals (Basel). 2023.
PMID: 38139850
Free PMC article.
Discovery of hydrazide-based pyridazino[4,5-b]indole scaffold as a new phosphoinositide 3-kinase (PI3K) inhibitor for breast cancer therapy.
Sarhan AAM, Boraei ATA, Barakat A, Nafie MS.
Sarhan AAM, et al.
RSC Adv. 2020 May 21;10(33):19534-19541. doi: 10.1039/d0ra02798g. eCollection 2020 May 20.
RSC Adv. 2020.
PMID: 35515454
Free PMC article.
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Expeditious Green Synthesis of Novel 4-Methyl-1,2,5,6-tetraazafluoranthen-3(2H)-one Analogue from Ninhydrin: N/S-Alkylation and Aza-Michael Addition.
Boraei ATA, Ghabbour HA, Sarhan AAM, Barakat A.
Boraei ATA, et al. Among authors: sarhan aam.
ACS Omega. 2020 Mar 3;5(10):5436-5442. doi: 10.1021/acsomega.0c00045. eCollection 2020 Mar 17.
ACS Omega. 2020.
PMID: 32201835
Free PMC article.
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Synthesis of a New Series of Nitrogen/Sulfur Heterocycles by Linking Four Rings: Indole; 1,2,4-Triazole; Pyridazine; and Quinoxaline.
Boraei ATA, Sarhan AAM, Yousuf S, Barakat A.
Boraei ATA, et al. Among authors: sarhan aam.
Molecules. 2020 Jan 21;25(3):450. doi: 10.3390/molecules25030450.
Molecules. 2020.
PMID: 31973234
Free PMC article.
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