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Assay platform for clinically relevant metallo-β-lactamases.
J Med Chem. 2013 Sep 12;56(17):6945-53. doi: 10.1021/jm400769b. Epub 2013 Aug 16.
J Med Chem. 2013.
PMID: 23898798
Free PMC article.
Chromophore-linked substrate (CLS405): probing metallo-β-lactamase activity and inhibition.
Makena A, van Berkel SS, Lejeune C, Owens RJ, Verma A, Salimraj R, Spencer J, Brem J, Schofield CJ.
Makena A, et al. Among authors: salimraj r.
ChemMedChem. 2013 Dec;8(12):1923-9. doi: 10.1002/cmdc.201300350. Epub 2013 Oct 25.
ChemMedChem. 2013.
PMID: 24166830
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Structural and Biochemical Characterization of Rm3, a Subclass B3 Metallo-β-Lactamase Identified from a Functional Metagenomic Study.
Salimraj R, Zhang L, Hinchliffe P, Wellington EM, Brem J, Schofield CJ, Gaze WH, Spencer J.
Salimraj R, et al.
Antimicrob Agents Chemother. 2016 Sep 23;60(10):5828-40. doi: 10.1128/AAC.00750-16. Print 2016 Oct.
Antimicrob Agents Chemother. 2016.
PMID: 27431213
Free PMC article.
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Crystal structures of VIM-1 complexes explain active site heterogeneity in VIM-class metallo-β-lactamases.
Salimraj R, Hinchliffe P, Kosmopoulou M, Tyrrell JM, Brem J, van Berkel SS, Verma A, Owens RJ, McDonough MA, Walsh TR, Schofield CJ, Spencer J.
Salimraj R, et al.
FEBS J. 2019 Jan;286(1):169-183. doi: 10.1111/febs.14695. Epub 2018 Nov 23.
FEBS J. 2019.
PMID: 30430727
Free PMC article.
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Structure-Guided Enhancement of Selectivity of Chemical Probe Inhibitors Targeting Bacterial Seryl-tRNA Synthetase.
Cain R, Salimraj R, Punekar AS, Bellini D, Fishwick CWG, Czaplewski L, Scott DJ, Harris G, Dowson CG, Lloyd AJ, Roper DI.
Cain R, et al. Among authors: salimraj r.
J Med Chem. 2019 Nov 14;62(21):9703-9717. doi: 10.1021/acs.jmedchem.9b01131. Epub 2019 Nov 5.
J Med Chem. 2019.
PMID: 31626547
Free article.
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Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1.
Wilding B, Pasqua AE, E A Chessum N, Pierrat OA, Hahner T, Tomlin K, Shehu E, Burke R, Richards GM, Whitton B, Arwert EN, Thapaliya A, Salimraj R, van Montfort R, Skawinska A, Hayes A, Raynaud F, Chopra R, Jones K, Newton G, Cheeseman MD.
Wilding B, et al. Among authors: salimraj r.
Bioorg Med Chem Lett. 2021 Jun 15;42:128050. doi: 10.1016/j.bmcl.2021.128050. Epub 2021 Apr 20.
Bioorg Med Chem Lett. 2021.
PMID: 33887439
Free PMC article.
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An evaluation of carcinogenicity predictors from short-term and sub chronic repeat-dose studies of agrochemicals in rats: Opportunities to refine and reduce animal use.
Mistry P, McInnes EF, Beevers C, Wolf D, Currie RA, Salimraj R, Parsons P.
Mistry P, et al. Among authors: salimraj r.
Toxicol Lett. 2021 Oct 15;351:18-27. doi: 10.1016/j.toxlet.2021.08.003. Epub 2021 Aug 5.
Toxicol Lett. 2021.
PMID: 34364947
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