Sadek B - Search Results

1

Repurposing SGLT2 Inhibitors for Neurological Disorders: A Focus on the Autism Spectrum Disorder.

Nakhal MM, Aburuz S, Sadek B, Akour A. Nakhal MM, et al. Among authors: sadek b. Molecules. 2022 Oct 23;27(21):7174. doi: 10.3390/molecules27217174. Molecules. 2022. PMID: 36364000 Free PMC article. Review.

2

Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H(3)-receptor antagonists.

Grassmann S, Sadek B, Ligneau X, Elz S, Ganellin CR, Arrang JM, Schwartz JC, Stark H, Schunack W. Grassmann S, et al. Among authors: sadek b. Eur J Pharm Sci. 2002 May;15(4):367-78. doi: 10.1016/s0928-0987(02)00024-6. Eur J Pharm Sci. 2002. PMID: 11988398

3

Novel histamine H(3)-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds.

Stark H, Sadek B, Krause M, Hüls A, Ligneau X, Ganellin CR, Arrang JM, Schwartz JC, Schunack W. Stark H, et al. Among authors: sadek b. J Med Chem. 2000 Oct 19;43(21):3987-94. doi: 10.1021/jm000966l. J Med Chem. 2000. PMID: 11052804

4

New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency.

Sasse A, Sadek B, Ligneau X, Elz S, Pertz HH, Luger P, Ganellin CR, Arrang JM, Schwartz JC, Schunack W, Stark H. Sasse A, et al. Among authors: sadek b. J Med Chem. 2000 Aug 24;43(17):3335-43. doi: 10.1021/jm000971p. J Med Chem. 2000. PMID: 10966752

5

Benzophenone derivatives and related compounds as potent histamine H3-receptor antagonists and potential PET/SPECT ligands.

Sasse A, Ligneau X, Sadek B, Elz S, Pertz HH, Ganellin CR, Arrang JM, Schwartz JC, Schunack W, Stark H. Sasse A, et al. Among authors: sadek b. Arch Pharm (Weinheim). 2001 Feb;334(2):45-52. doi: 10.1002/1521-4184(200102)334:2<45::aid-ardp45>3.0.co;2-2. Arch Pharm (Weinheim). 2001. PMID: 11268774

6

Analogues and derivatives of ciproxifan, a novel prototype for generating potent histamine H3-receptor antagonists.

Stark H, Ligneau X, Sadek B, Ganellin CR, Arrang JM, Schwartz JC, Schunack W. Stark H, et al. Among authors: sadek b. Bioorg Med Chem Lett. 2000 Oct 16;10(20):2379-82. doi: 10.1016/s0960-894x(00)00473-x. Bioorg Med Chem Lett. 2000. PMID: 11055360

7

Novel N-phenylcarbamothioylbenzamides with anti-inflammatory activity and prostaglandin E2 inhibitory properties.

Limban C, Missir AV, Fahelelbom KM, Al-Tabakha MM, Caproiu MT, Sadek B. Limban C, et al. Among authors: sadek b. Drug Des Devel Ther. 2013 Aug 28;7:883-92. doi: 10.2147/DDDT.S46691. eCollection 2013. Drug Des Devel Ther. 2013. PMID: 24039398 Free PMC article.

8

The Neuroprotective Effects of Histamine H3 Receptor Antagonist E177 on Pilocarpine-Induced Status Epilepticus in Rats.

Alachkar A, Azimullah S, Ojha SK, Beiram R, Łażewska D, Kieć-Kononowicz K, Sadek B. Alachkar A, et al. Among authors: sadek b. Molecules. 2019 Nov 14;24(22):4106. doi: 10.3390/molecules24224106. Molecules. 2019. PMID: 31739417 Free PMC article.

9

Antagonism of Histamine H3 receptors Alleviates Pentylenetetrazole-Induced Kindling and Associated Memory Deficits by Mitigating Oxidative Stress, Central Neurotransmitters, and c-Fos Protein Expression in Rats.

Alachkar A, Azimullah S, Lotfy M, Adeghate E, Ojha SK, Beiram R, Łażewska D, Kieć-Kononowicz K, Sadek B. Alachkar A, et al. Among authors: sadek b. Molecules. 2020 Mar 30;25(7):1575. doi: 10.3390/molecules25071575. Molecules. 2020. PMID: 32235506 Free PMC article.

10

The Multi-Targeting Ligand ST-2223 with Histamine H₃ Receptor and Dopamine D₂/D₃ Receptor Antagonist Properties Mitigates Autism-Like Repetitive Behaviors and Brain Oxidative Stress in Mice.

Eissa N, Venkatachalam K, Jayaprakash P, Falkenstein M, Dubiel M, Frank A, Reiner-Link D, Stark H, Sadek B. Eissa N, et al. Among authors: sadek b. Int J Mol Sci. 2021 Feb 16;22(4):1947. doi: 10.3390/ijms22041947. Int J Mol Sci. 2021. PMID: 33669336 Free PMC article.

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