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Synthesis and in Vitro Screening of New Series of 2,6-Dipeptidyl-anthraquinones: Influence of Side Chain Length on HIV-1 Nucleocapsid Inhibitors.
Frecentese F, Sosic A, Saccone I, Gamba E, Link K, Miola A, Cappellini M, Cattelan MG, Severino B, Fiorino F, Magli E, Corvino A, Perissutti E, Fabris D, Gatto B, Caliendo G, Santagada V. Frecentese F, et al. Among authors: saccone i. J Med Chem. 2016 Mar 10;59(5):1914-24. doi: 10.1021/acs.jmedchem.5b01494. Epub 2016 Feb 3. J Med Chem. 2016. PMID: 26797100
New 5-HT1A, 5HT2A and 5HT2C receptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation.
Fiorino F, Magli E, Kędzierska E, Ciano A, Corvino A, Severino B, Perissutti E, Frecentese F, Di Vaio P, Saccone I, Izzo AA, Capasso R, Massarelli P, Rossi I, Orzelska-Gòrka J, Kotlińska JH, Santagada V, Caliendo G. Fiorino F, et al. Among authors: saccone i. Bioorg Med Chem. 2017 Oct 15;25(20):5820-5837. doi: 10.1016/j.bmc.2017.09.018. Epub 2017 Sep 18. Bioorg Med Chem. 2017. PMID: 28943244
1,2,4-Thiadiazolidin-3,5-diones as novel hydrogen sulfide donors.
Severino B, Corvino A, Fiorino F, Luciano P, Frecentese F, Magli E, Saccone I, Di Vaio P, Citi V, Calderone V, Servillo L, Casale R, Cirino G, Vellecco V, Bucci M, Perissutti E, Santagada V, Caliendo G. Severino B, et al. Among authors: saccone i. Eur J Med Chem. 2018 Jan 1;143:1677-1686. doi: 10.1016/j.ejmech.2017.10.068. Epub 2017 Nov 11. Eur J Med Chem. 2018. PMID: 29133036
Non-Natural Linker Configuration in 2,6-Dipeptidyl-Anthraquinones Enhances the Inhibition of TAR RNA Binding/Annealing Activities by HIV-1 NC and Tat Proteins.
Sosic A, Saccone I, Carraro C, Kenderdine T, Gamba E, Caliendo G, Corvino A, Di Vaio P, Fiorino F, Magli E, Perissutti E, Santagada V, Severino B, Spada V, Fabris D, Frecentese F, Gatto B. Sosic A, et al. Among authors: saccone i. Bioconjug Chem. 2018 Jul 18;29(7):2195-2207. doi: 10.1021/acs.bioconjchem.8b00104. Epub 2018 Jun 12. Bioconjug Chem. 2018. PMID: 29791798 Free PMC article.
Synthesis, docking studies, and pharmacological evaluation of 5HT2C ligands containing the N'-cyanoisonicotinamidine or N'-cyanopicolinamidine nucleus.
Magli E, Kędzierska E, Kaczor AA, Severino B, Corvino A, Perissutti E, Frecentese F, Saccone I, Massarelli P, Gibuła-Tarłowska E, Kotlińska JH, Santagada V, Caliendo G, Fiorino F. Magli E, et al. Among authors: saccone i. Arch Pharm (Weinheim). 2019 May;352(5):e1800373. doi: 10.1002/ardp.201800373. Epub 2019 Apr 26. Arch Pharm (Weinheim). 2019. PMID: 31025433
18 results