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Deactivatable Bisubstrate Inhibitors of Protein Kinases.
Molecules. 2022 Oct 8;27(19):6689. doi: 10.3390/molecules27196689.
Molecules. 2022.
PMID: 36235226
Free PMC article.
Conjugates of adenosine mimetics and arginine-rich peptides serve as inhibitors and fluorescent probes but not as long-lifetime photoluminescent probes for protein arginine methyltransferases.
Lavogina D, Nasirova N, Sõrmus T, Tähtjärv T, Enkvist E, Viht K, Haljasorg T, Herodes K, Jaal J, Uri A.
Lavogina D, et al. Among authors: sormus t.
J Pept Sci. 2023 Mar;29(3):e3456. doi: 10.1002/psc.3456. Epub 2022 Oct 28.
J Pept Sci. 2023.
PMID: 36208424
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Construction of Covalent Bisubstrate Inhibitor of Protein Kinase Reacting with Cysteine Residue at Substrate-Binding Site.
Sõrmus T, Lavogina D, Teearu A, Enkvist E, Uri A, Viht K.
Sõrmus T, et al.
J Med Chem. 2022 Aug 25;65(16):10975-10991. doi: 10.1021/acs.jmedchem.2c00067. Epub 2022 Aug 12.
J Med Chem. 2022.
PMID: 35960538
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Efficient photocaging of a tight-binding bisubstrate inhibitor of cAMP-dependent protein kinase.
Sõrmus T, Lavogina D, Enkvist E, Uri A, Viht K.
Sõrmus T, et al.
Chem Commun (Camb). 2019 Sep 21;55(74):11147-11150. doi: 10.1039/c9cc04978a. Epub 2019 Aug 29.
Chem Commun (Camb). 2019.
PMID: 31464306
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