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Year | Number of Results |
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2021 | 1 |
2022 | 1 |
2023 | 1 |
2024 | 1 |
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Covalent Fragment Screening and Optimization Identifies the Chloroacetohydrazide Scaffold as Inhibitors for Ubiquitin C-terminal Hydrolase L1.
J Med Chem. 2024 Mar 28;67(6):4496-4524. doi: 10.1021/acs.jmedchem.3c01661. Epub 2024 Mar 15.
J Med Chem. 2024.
PMID: 38488146
Identification of covalent fragment inhibitors for Plasmodium falciparum UCHL3 with anti-malarial efficacy.
Imhoff RD, Rosenthal MR, Ashraf K, Bhanot P, Ng CL, Flaherty DP.
Imhoff RD, et al.
Bioorg Med Chem Lett. 2023 Oct 1;94:129458. doi: 10.1016/j.bmcl.2023.129458. Epub 2023 Aug 25.
Bioorg Med Chem Lett. 2023.
PMID: 37634761
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Structure-activity relationship studies for inhibitors for vancomycin-resistant Enterococcus and human carbonic anhydrases.
An W, Holly KJ, Nocentini A, Imhoff RD, Hewitt CS, Abutaleb NS, Cao X, Seleem MN, Supuran CT, Flaherty DP.
An W, et al. Among authors: imhoff rd.
J Enzyme Inhib Med Chem. 2022 Dec;37(1):1838-1844. doi: 10.1080/14756366.2022.2092729.
J Enzyme Inhib Med Chem. 2022.
PMID: 35758212
Free PMC article.
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Optimization and Anti-Cancer Properties of Fluoromethylketones as Covalent Inhibitors for Ubiquitin C-Terminal Hydrolase L1.
Krabill AD, Chen H, Hussain S, Hewitt CS, Imhoff RD, Muli CS, Das C, Galardy PJ, Wendt MK, Flaherty DP.
Krabill AD, et al. Among authors: imhoff rd.
Molecules. 2021 Feb 25;26(5):1227. doi: 10.3390/molecules26051227.
Molecules. 2021.
PMID: 33668938
Free PMC article.
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