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Synthesis, biological evaluation and in silico modeling of novel pan-genotypic NS5A inhibitors.
Bioorg Med Chem. 2020 Oct 15;28(20):115716. doi: 10.1016/j.bmc.2020.115716. Epub 2020 Aug 20.
Bioorg Med Chem. 2020.
PMID: 33069072
Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses.
Ivashchenko AA, Mitkin OD, Jones JC, Nikitin AV, Koryakova AG, Ryakhovskiy A, Karapetian RN, Kravchenko DV, Aladinskiy V, Leneva IA, Falynskova IN, Glubokova EA, Govorkova EA, Ivachtchenko AV.
Ivashchenko AA, et al. Among authors: ryakhovskiy a.
J Med Chem. 2020 Sep 10;63(17):9403-9420. doi: 10.1021/acs.jmedchem.0c00565. Epub 2020 Aug 17.
J Med Chem. 2020.
PMID: 32787099
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Synthesis, inhibitory activity and oral dosing formulation of AV5124, the structural analogue of influenza virus endonuclease inhibitor baloxavir.
Ivashchenko AA, Mitkin OD, Jones JC, Nikitin AV, Koryakova AG, Karapetian RN, Kravchenko DV, Mochalov SV, Ryakhovskiy AA, Aladinskiy V, Leneva IA, Falynskova IN, Glubokova EA, Govorkova EA, Ivachtchenko AV.
Ivashchenko AA, et al. Among authors: ryakhovskiy aa.
J Antimicrob Chemother. 2021 Mar 12;76(4):1010-1018. doi: 10.1093/jac/dkaa524.
J Antimicrob Chemother. 2021.
PMID: 33367751
Free PMC article.
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Optimization of a cellular HBV infection model for use in high-throughput drug screening.
Kartashova NP, Iarovenko SI, Glubokova EA, Potemkin IA, Karlsen AA, Leneva IA, Kyuregyan KK, Ryakhovskiy AA, Mikhailov MI.
Kartashova NP, et al. Among authors: ryakhovskiy aa.
Acta Virol. 2021;65(1):82-88. doi: 10.4149/av_2021_110.
Acta Virol. 2021.
PMID: 33827225
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Exploring bioactivity potential of polyphenolic water-soluble lignin derivative.
Fedoros EI, Baldueva IA, Perminova IV, Badun GA, Chernysheva MG, Grozdova ID, Melik-Nubarov NS, Danilova AB, Nekhaeva TL, Kuznetsova AI, Emelyanova NV, Ryakhovskiy AA, Pigarev SE, Semenov AL, Tyndyk ML, Gubareva EA, Panchenko AV, Bykov VN, Anisimov VN.
Fedoros EI, et al. Among authors: ryakhovskiy aa.
Environ Res. 2020 Dec;191:110049. doi: 10.1016/j.envres.2020.110049. Epub 2020 Sep 11.
Environ Res. 2020.
PMID: 32926891
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S/MAR and TRE can be found co-localized within regulatory chromosome regions of some tissue-specifically expressed genes of Drosophila melanogaster.
Ryakhovskiy AA, Tillib SV.
Ryakhovskiy AA, et al.
Dokl Biochem Biophys. 2007 Sep-Oct;416:264-7. doi: 10.1134/s1607672907050109.
Dokl Biochem Biophys. 2007.
PMID: 18064828
No abstract available.
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