Ruiu S - Search Results

1

Novel pyrazole derivatives as neutral CB₁ antagonists with significant activity towards food intake.

Manca I, Mastinu A, Olimpieri F, Falzoi M, Sani M, Ruiu S, Loriga G, Volonterio A, Tambaro S, Bottazzi ME, Zanda M, Pinna GA, Lazzari P. Manca I, et al. Among authors: ruiu s. Eur J Med Chem. 2013 Apr;62:256-69. doi: 10.1016/j.ejmech.2012.12.056. Epub 2013 Jan 11. Eur J Med Chem. 2013. PMID: 23357307

2

N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as mu-opioid receptor agonists. Effects on mu-affinity of arylalkenyl chain modifications.

Pinna GA, Cignarella G, Loriga G, Murineddu G, Mussinu JM, Ruiu S, Fadda P, Fratta W. Pinna GA, et al. Among authors: ruiu s. Bioorg Med Chem. 2002 Jun;10(6):1929-37. doi: 10.1016/s0968-0896(01)00436-9. Bioorg Med Chem. 2002. PMID: 11937351

3

Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors.

Mussinu JM, Ruiu S, Mulè AC, Pau A, Carai MA, Loriga G, Murineddu G, Pinna GA. Mussinu JM, et al. Among authors: ruiu s. Bioorg Med Chem. 2003 Jan 17;11(2):251-63. doi: 10.1016/s0968-0896(02)00319-x. Bioorg Med Chem. 2003. PMID: 12470719

4

Synthesis and characterization of NESS 0327: a novel putative antagonist of the CB1 cannabinoid receptor.

Ruiu S, Pinna GA, Marchese G, Mussinu JM, Saba P, Tambaro S, Casti P, Vargiu R, Pani L. Ruiu S, et al. J Pharmacol Exp Ther. 2003 Jul;306(1):363-70. doi: 10.1124/jpet.103.049924. Epub 2003 Mar 27. J Pharmacol Exp Ther. 2003. PMID: 12663689

5

Synthesis of novel diazatricyclodecanes (DTDs). Effects of structural variation at the C3' allyl end and at the phenyl ring of the cinnamyl chain on mu-receptor affinity and opioid antinociception.

Pinna GA, Cignarella G, Ruiu S, Loriga G, Murineddu G, Villa S, Grella GE, Cossu G, Fratta W. Pinna GA, et al. Among authors: ruiu s. Bioorg Med Chem. 2003 Sep 1;11(18):4015-26. doi: 10.1016/s0968-0896(03)00373-0. Bioorg Med Chem. 2003. PMID: 12927864

6

Haloperidol versus risperidone on rat "early onset" vacuous chewing.

Marchese G, Bartholini F, Casu MA, Ruiu S, Casti P, Congeddu E, Tambaro S, Pani L. Marchese G, et al. Among authors: ruiu s. Behav Brain Res. 2004 Feb 4;149(1):9-16. doi: 10.1016/s0166-4328(03)00192-x. Behav Brain Res. 2004. PMID: 14739005

7

Evaluation of tamsulosin and alfuzosin activity in the rat vas deferens: relevance to ejaculation delays.

Tambaro S, Ruiu S, Dessi C, Mongeau R, Marchese G, Pani L. Tambaro S, et al. Among authors: ruiu s. J Pharmacol Exp Ther. 2005 Feb;312(2):710-7. doi: 10.1124/jpet.104.074740. Epub 2004 Oct 6. J Pharmacol Exp Ther. 2005. PMID: 15470085

8

Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzo[g]indazole-based ligands for cannabinoid receptors.

Murineddu G, Ruiu S, Mussinu JM, Loriga G, Grella GE, Carai MA, Lazzari P, Pani L, Pinna GA. Murineddu G, et al. Among authors: ruiu s. Bioorg Med Chem. 2005 May 2;13(9):3309-20. doi: 10.1016/j.bmc.2005.02.032. Bioorg Med Chem. 2005. PMID: 15809166

9

Modulation of ATP-mediated contractions of the rat vas deferens through presynaptic cannabinoid receptors.

Tambaro S, Mongeau R, Dessi C, Pani L, Ruiu S. Tambaro S, et al. Among authors: ruiu s. Eur J Pharmacol. 2005 Nov 21;525(1-3):150-3. doi: 10.1016/j.ejphar.2005.09.058. Epub 2005 Nov 3. Eur J Pharmacol. 2005. PMID: 16271359

10

Tricyclic pyrazoles. 3. Synthesis, biological evaluation, and molecular modeling of analogues of the cannabinoid antagonist 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide.

Murineddu G, Ruiu S, Loriga G, Manca I, Lazzari P, Reali R, Pani L, Toma L, Pinna GA. Murineddu G, et al. Among authors: ruiu s. J Med Chem. 2005 Nov 17;48(23):7351-62. doi: 10.1021/jm050317f. J Med Chem. 2005. PMID: 16279795

A series of analogues of 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 4a (NESS 0327) (Ruiu, S.; Pinna, G. A.; Marchese, G.; Mussinu, J. M.; Saba, P.; Tambaro, S.; Casti, P.; Vargiu, R.; …

A series of analogues of 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxam …

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