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Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals.
Burgart YV, Elkina NA, Shchegolkov EV, Krasnykh OP, Makhaeva GF, Triandafilova GA, Solodnikov SY, Boltneva NP, Rudakova EV, Kovaleva NV, Serebryakova OG, Ulitko MV, Borisevich SS, Gerasimova NA, Evstigneeva NP, Kozlov SA, Korolkova YV, Minin AS, Belousova AV, Mozhaitsev ES, Klabukov AM, Saloutin VI. Burgart YV, et al. Among authors: rudakova ev. Molecules. 2022 Dec 21;28(1):59. doi: 10.3390/molecules28010059. Molecules. 2022. PMID: 36615256 Free PMC article.
A new selective inhibitor of mouse blood plasma carboxylesterase.
Rudakova EV, Makhaeva GF, Galenko TG, Aksinenko AY, Sokolov VB, Martynov IV. Rudakova EV, et al. Dokl Biochem Biophys. 2013 Mar-Apr;449:87-9. doi: 10.1134/S1607672913020099. Epub 2013 May 9. Dokl Biochem Biophys. 2013. PMID: 23657654 No abstract available.
Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors.
Shchegol'kov EV, Makhaeva GF, Boltneva NP, Lushchekina SV, Serebryakova OG, Rudakova EV, Kovaleva NV, Burgart YV, Saloutin VI, Chupakhin ON, Bachurin SO, Richardson RJ. Shchegol'kov EV, et al. Among authors: rudakova ev. Bioorg Med Chem. 2017 Aug 1;25(15):3997-4007. doi: 10.1016/j.bmc.2017.05.045. Epub 2017 May 20. Bioorg Med Chem. 2017. PMID: 28578994
44 results