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RS6077 induces mitotic arrest and selectively activates cell death in human cancer cell lines and in a lymphoma tumor in vivo.
Eur J Med Chem. 2023 Jan 15;246:114997. doi: 10.1016/j.ejmech.2022.114997. Epub 2022 Dec 5.
Eur J Med Chem. 2023.
PMID: 36502578
Reverse transcriptase inhibitors promote the remodelling of nuclear architecture and induce autophagy in prostate cancer cells.
Bellisai C, Sciamanna I, Rovella P, Giovannini D, Baranzini M, Pugliese GM, Zeya Ansari MS, Milite C, Sinibaldi-Vallebona P, Cirilli R, Sbardella G, Pichierri P, Trisciuoglio D, Lavia P, Serafino A, Spadafora C.
Bellisai C, et al. Among authors: rovella p.
Cancer Lett. 2020 May 28;478:133-145. doi: 10.1016/j.canlet.2020.02.029. Epub 2020 Feb 26.
Cancer Lett. 2020.
PMID: 32112906
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Importin-β/karyopherin-β1 modulates mitotic microtubule function and taxane sensitivity in cancer cells via its nucleoporin-binding region.
Verrico A, Rovella P, Di Francesco L, Damizia M, Staid DS, Le Pera L, Schininà ME, Lavia P.
Verrico A, et al. Among authors: rovella p.
Oncogene. 2020 Jan;39(2):454-468. doi: 10.1038/s41388-019-0989-x. Epub 2019 Sep 6.
Oncogene. 2020.
PMID: 31492900
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New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors.
La Regina G, Bai R, Coluccia A, Naccarato V, Famiglini V, Nalli M, Masci D, Verrico A, Rovella P, Mazzoccoli C, Da Pozzo E, Cavallini C, Martini C, Vultaggio S, Dondio G, Varasi M, Mercurio C, Hamel E, Lavia P, Silvestri R.
La Regina G, et al. Among authors: rovella p.
Eur J Med Chem. 2018 May 25;152:283-297. doi: 10.1016/j.ejmech.2018.04.042. Epub 2018 Apr 25.
Eur J Med Chem. 2018.
PMID: 29730191
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Visualization of human karyopherin beta-1/importin beta-1 interactions with protein partners in mitotic cells by co-immunoprecipitation and proximity ligation assays.
Di Francesco L, Verrico A, Asteriti IA, Rovella P, Cirigliano P, Guarguaglini G, Schininà ME, Lavia P.
Di Francesco L, et al. Among authors: rovella p.
Sci Rep. 2018 Jan 30;8(1):1850. doi: 10.1038/s41598-018-19351-9.
Sci Rep. 2018.
PMID: 29382863
Free PMC article.
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Mitotic cell death induction by targeting the mitotic spindle with tubulin-inhibitory indole derivative molecules.
Di Cesare E, Verrico A, Miele A, Giubettini M, Rovella P, Coluccia A, Famiglini V, La Regina G, Cundari E, Silvestri R, Lavia P.
Di Cesare E, et al. Among authors: rovella p.
Oncotarget. 2017 Mar 21;8(12):19738-19759. doi: 10.18632/oncotarget.14980.
Oncotarget. 2017.
PMID: 28160569
Free PMC article.
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