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Identification of a Potent and Selective 5-HT1A Receptor Agonist with In Vitro and In Vivo Antinociceptive Activity.
Linciano P, Sorbi C, Comitato A, Lesniak A, Bujalska-Zadrożny M, Pawłowska A, Bielenica A, Orzelska-Górka J, Kędzierska E, Biała G, Ronsisvalle S, Limoncella S, Casarini L, Cichero E, Fossa P, Satała G, Bojarski AJ, Brasili L, Bardoni R, Franchini S. Linciano P, et al. Among authors: ronsisvalle s. ACS Chem Neurosci. 2020 Dec 16;11(24):4111-4127. doi: 10.1021/acschemneuro.0c00289. Epub 2020 Dec 2. ACS Chem Neurosci. 2020. PMID: 33263393 Free PMC article.
Novel potent and selective σ ligands: evaluation of their agonist and antagonist properties.
Marrazzo A, Cobos EJ, Parenti C, Aricò G, Marrazzo G, Ronsisvalle S, Pasquinucci L, Prezzavento O, Colabufo NA, Contino M, González LG, Scoto GM, Ronsisvalle G. Marrazzo A, et al. Among authors: ronsisvalle g, ronsisvalle s. J Med Chem. 2011 May 26;54(10):3669-73. doi: 10.1021/jm200144j. Epub 2011 Apr 21. J Med Chem. 2011. PMID: 21476493
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives.
Franchini S, Battisti UM, Prandi A, Tait A, Borsari C, Cichero E, Fossa P, Cilia A, Prezzavento O, Ronsisvalle S, Aricò G, Parenti C, Brasili L. Franchini S, et al. Among authors: ronsisvalle s. Eur J Med Chem. 2016 Apr 13;112:1-19. doi: 10.1016/j.ejmech.2016.01.059. Epub 2016 Feb 1. Eur J Med Chem. 2016. PMID: 26874044 Free article.
Synthesis, biological evaluation and molecular modeling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT1A receptor agonists.
Franchini S, Manasieva LI, Sorbi C, Battisti UM, Fossa P, Cichero E, Denora N, Iacobazzi RM, Cilia A, Pirona L, Ronsisvalle S, Aricò G, Brasili L. Franchini S, et al. Among authors: ronsisvalle s. Eur J Med Chem. 2017 Jan 5;125:435-452. doi: 10.1016/j.ejmech.2016.09.050. Epub 2016 Sep 17. Eur J Med Chem. 2017. PMID: 27689727 Free article.
Structure-Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma.
Franchini S, Sorbi C, Battisti UM, Tait A, Bencheva LI, Cichero E, Fossa P, Cilia A, Prezzavento O, Ronsisvalle S, Aricò G, Benassi L, Vaschieri C, Azzoni P, Magnoni C, Brasili L. Franchini S, et al. Among authors: ronsisvalle s. ChemMedChem. 2017 Nov 22;12(22):1893-1905. doi: 10.1002/cmdc.201700427. Epub 2017 Oct 30. ChemMedChem. 2017. PMID: 28940806 Free article.
Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT1A receptor agonists for CNS disorders and neuropathic pain.
Franchini S, Bencheva LI, Battisti UM, Tait A, Sorbi C, Fossa P, Cichero E, Ronsisvalle S, Aricò G, Denora N, Iacobazzi RM, Cilia A, Pirona L, Brasili L. Franchini S, et al. Among authors: ronsisvalle s. Future Med Chem. 2018 Sep 1;10(18):2137-2154. doi: 10.4155/fmc-2018-0107. Epub 2018 Jul 25. Future Med Chem. 2018. PMID: 30043643
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity.
Franchini S, Sorbi C, Linciano P, Carnevale G, Tait A, Ronsisvalle S, Buccioni M, Del Bello F, Cilia A, Pirona L, Denora N, Iacobazzi RM, Brasili L. Franchini S, et al. Among authors: ronsisvalle s. Eur J Med Chem. 2019 Aug 15;176:310-325. doi: 10.1016/j.ejmech.2019.05.024. Epub 2019 May 11. Eur J Med Chem. 2019. PMID: 31112892
BS148 Reduces the Aggressiveness of Metastatic Melanoma via Sigma-2 Receptor Targeting.
Sorbi C, Belluti S, Atene CG, Marocchi F, Linciano P, Roy N, Paradiso E, Casarini L, Ronsisvalle S, Zanocco-Marani T, Brasili L, Lanfrancone L, Imbriano C, Di Rocco G, Franchini S. Sorbi C, et al. Among authors: ronsisvalle s. Int J Mol Sci. 2023 Jun 2;24(11):9684. doi: 10.3390/ijms24119684. Int J Mol Sci. 2023. PMID: 37298633 Free PMC article.
72 results