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Discovery and Optimization of Indoline-Based Compounds as Dual 5-LOX/sEH Inhibitors: In Vitro and In Vivo Anti-Inflammatory Characterization.
Cerqua I, Musella S, Peltner LK, D'Avino D, Di Sarno V, Granato E, Vestuto V, Di Matteo R, Pace S, Ciaglia T, Bilancia R, Smaldone G, Di Matteo F, Di Micco S, Bifulco G, Pepe G, Basilicata MG, Rodriquez M, Gomez-Monterrey IM, Campiglia P, Ostacolo C, Roviezzo F, Werz O, Rossi A, Bertamino A. Cerqua I, et al. Among authors: rodriquez m. J Med Chem. 2022 Nov 10;65(21):14456-14480. doi: 10.1021/acs.jmedchem.2c00817. Epub 2022 Nov 1. J Med Chem. 2022. PMID: 36318728 Free PMC article.
Salicylic Acid Release from Syndiotactic Polystyrene Staple Fibers.
Covelli V, Cozzolino A, Rizzo P, Rodriquez M, Vestuto V, Bertamino A, Daniel C, Guerra G. Covelli V, et al. Among authors: rodriquez m. Molecules. 2023 Jun 29;28(13):5095. doi: 10.3390/molecules28135095. Molecules. 2023. PMID: 37446756 Free PMC article.
Towards an Improvement of Anticancer Activity of Benzyl Adenosine Analogs.
Covelli V, Grimaldi M, Randino R, Firoznezhad M, Proto MC, Simone V, Matteoli G, Gazzerro P, Bifulco M, D'Ursi AM, Rodriquez M. Covelli V, et al. Among authors: rodriquez m. Molecules. 2021 Nov 25;26(23):7146. doi: 10.3390/molecules26237146. Molecules. 2021. PMID: 34885721 Free PMC article.
Benzodiazepine Scaffold as Drug-like Molecular Simplification of FR235222: A Chemical Tool for Exploring HDAC Inhibition.
Randino R, Moronese I, Cini E, Bizzarro V, Persico M, Grimaldi M, Scrima M, D'Ursi AM, Novellino E, Sobarzo-Sanchez E, Rastrelli L, Fattorusso C, Petrella A, Rodriquez M, Taddei M. Randino R, et al. Among authors: rodriquez m. Curr Top Med Chem. 2017;17(4):441-459. doi: 10.2174/1568026616666160824105645. Curr Top Med Chem. 2017. PMID: 27558677
126 results