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Leishmanicidal activity and 4D quantitative structure-activity relationship and molecular docking studies of vanillin-containing 1,2,3-triazole derivatives.
Rodrigues Gazolla PA, Lima WP, de Aguiar AR, Gonçalves Borsodi MP, Costa AV, de Oliveira FM, de Oliveira OV, Andreazza Costa MC, Castro Ferreira MM, do Nascimento CJ, Junker J, Vaz BG, Teixeira RR. Rodrigues Gazolla PA, et al. Future Med Chem. 2024 Jan;16(2):139-155. doi: 10.4155/fmc-2023-0246. Epub 2023 Dec 22. Future Med Chem. 2024. PMID: 38131191
Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors.
Maltarollo VG, da Silva EB, Kronenberger T, Sena Andrade MM, de Lima Marques GV, Cândido Oliveira NJ, Santos LH, Oliveira Rezende Júnior C, Cassiano Martinho AC, Skinner D, Fajtová P, M Fernandes TH, Silveira Dos Santos ED, Rodrigues Gazolla PA, Martins de Souza AP, da Silva ML, Dos Santos FS, Lavorato SN, Oliveira Bretas AC, Carvalho DT, Franco LL, Luedtke S, Giardini MA, Poso A, Dias LC, Podust LM, Alves RJ, McKerrow J, Andrade SF, Teixeira RR, Siqueira-Neto JL, O'Donoghue A, de Oliveira RB, Ferreira RS. Maltarollo VG, et al. Among authors: rodrigues gazolla pa. Future Med Chem. 2023 Jun;15(11):959-985. doi: 10.4155/fmc-2023-0034. Epub 2023 Jul 12. Future Med Chem. 2023. PMID: 37435731
Synthesis and virucide activity on zika virus of 1,2,3-triazole-containing vanillin derivatives.
da Silva Rodrigues JV, Rodrigues Gazolla PA, da Cruz Pereira I, Dias RS, Poly da Silva IE, Oliveira Prates JW, de Souza Gomes I, de Azevedo Silveira S, Costa AV, de Oliveira FM, de Aguiar AR, Canedo da Silva C, Teixeira RR, de Paula SO. da Silva Rodrigues JV, et al. Among authors: rodrigues gazolla pa. Antiviral Res. 2023 Apr;212:105578. doi: 10.1016/j.antiviral.2023.105578. Epub 2023 Mar 17. Antiviral Res. 2023. PMID: 36934985
Eugenol derivatives with 1,2,3-triazole moieties: Oral treatment of cutaneous leishmaniasis and a quantitative structure-activity relationship model for their leishmanicidal activity.
Teixeira RR, Rodrigues Gazolla PA, Borsodi MPG, Castro Ferreira MM, Andreazza Costa MC, Costa AV, Cabral Abreu Grijó B, Rossi Bergmann B, Lima WP. Teixeira RR, et al. Among authors: rodrigues gazolla pa. Exp Parasitol. 2022 Jul;238:108269. doi: 10.1016/j.exppara.2022.108269. Epub 2022 May 5. Exp Parasitol. 2022. PMID: 35526574