Rodeschini V - Search Results

1

Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action.

Fernández-Montalván AE, Berger M, Kuropka B, Koo SJ, Badock V, Weiske J, Puetter V, Holton SJ, Stöckigt D, Ter Laak A, Centrella PA, Clark MA, Dumelin CE, Sigel EA, Soutter HH, Troast DM, Zhang Y, Cuozzo JW, Keefe AD, Roche D, Rodeschini V, Chaikuad A, Díaz-Sáez L, Bennett JM, Fedorov O, Huber KVM, Hübner J, Weinmann H, Hartung IV, Gorjánácz M. Fernández-Montalván AE, et al. Among authors: rodeschini v. ACS Chem Biol. 2017 Nov 17;12(11):2730-2736. doi: 10.1021/acschembio.7b00708. Epub 2017 Oct 24. ACS Chem Biol. 2017. PMID: 29043777 Free PMC article.

2

New Caspase-1 inhibitor by scaffold hopping into bio-inspired 3D-fragment space.

Brethon A, Chantalat L, Christin O, Clary L, Fournier JF, Gastreich M, Harris CS, Isabet T, Pascau J, Thoreau E, Roche D, Rodeschini V. Brethon A, et al. Among authors: rodeschini v. Bioorg Med Chem Lett. 2017 Dec 15;27(24):5373-5377. doi: 10.1016/j.bmcl.2017.11.015. Epub 2017 Nov 9. Bioorg Med Chem Lett. 2017. PMID: 29157864

3

Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne.

Fournier JF, Clary L, Chambon S, Dumais L, Harris CS, Millois C, Pierre R, Talano S, Thoreau É, Aubert J, Aurelly M, Bouix-Peter C, Brethon A, Chantalat L, Christin O, Comino C, El-Bazbouz G, Ghilini AL, Isabet T, Lardy C, Luzy AP, Mathieu C, Mebrouk K, Orfila D, Pascau J, Reverse K, Roche D, Rodeschini V, Hennequin LF. Fournier JF, et al. Among authors: rodeschini v. J Med Chem. 2018 May 10;61(9):4030-4051. doi: 10.1021/acs.jmedchem.8b00067. Epub 2018 Apr 24. J Med Chem. 2018. PMID: 29648825

4

Comparison of the cytotoxic effects of enantiopure PPAPs, including nemorosone and clusianone.

Simpkins NS, Holtrup F, Rodeschini V, Taylor JD, Wolf R. Simpkins NS, et al. Among authors: rodeschini v. Bioorg Med Chem Lett. 2012 Oct 1;22(19):6144-7. doi: 10.1016/j.bmcl.2012.08.023. Epub 2012 Aug 11. Bioorg Med Chem Lett. 2012. PMID: 22944119

5

Synthesis of (+/-)-clusianone: high-yielding bridgehead and diketone substitutions by regioselective lithiation of enol ether derivatives of bicyclo[3.3.1]nonane-2,4,9-triones.

Rodeschini V, Ahmad NM, Simpkins NS. Rodeschini V, et al. Org Lett. 2006 Nov 9;8(23):5283-5. doi: 10.1021/ol0620592. Org Lett. 2006. PMID: 17078698

6

Kinetic resolution in a bridgehead lithiation mediated by a chiral bis-lithium amide: assignment of the absolute configuration of clusianone.

Rodeschini V, Simpkins NS, Wilson C. Rodeschini V, et al. J Org Chem. 2007 May 25;72(11):4265-7. doi: 10.1021/jo070225t. Epub 2007 Apr 28. J Org Chem. 2007. PMID: 17465570

7

Synthesis of polyprenylated acylphloroglucinols using bridgehead lithiation: the total synthesis of racemic clusianone and a formal synthesis of racemic garsubellin A.

Ahmad NM, Rodeschini V, Simpkins NS, Ward SE, Blake AJ. Ahmad NM, et al. Among authors: rodeschini v. J Org Chem. 2007 Jun 22;72(13):4803-15. doi: 10.1021/jo070388h. Epub 2007 May 26. J Org Chem. 2007. PMID: 17530804

8

Synthetic studies towards garsubellin A: synthesis of model systems and potential mimics by regioselective lithiation of bicyclo[3.3.1]nonane-2,4,9-trione derivatives from catechinic acid.

Ahmad NM, Rodeschini V, Simpkins NS, Ward SE, Wilson C. Ahmad NM, et al. Among authors: rodeschini v. Org Biomol Chem. 2007 Jun 21;5(12):1924-34. doi: 10.1039/b704311b. Epub 2007 May 15. Org Biomol Chem. 2007. PMID: 17551642

9

Enantioselective approaches to potential MetAP-2 reversible inhibitors.

Rodeschini V, Van de Weghe P, Salomon E, Tarnus C, Eustache J. Rodeschini V, et al. J Org Chem. 2005 Mar 18;70(6):2409-12. doi: 10.1021/jo047858h. J Org Chem. 2005. PMID: 15760245

10

MetAP-2 inhibitors based on the fumagillin structure. Side-chain modification and ring-substituted analogues.

Rodeschini V, Boiteau JG, Van de Weghe P, Tarnus C, Eustache J. Rodeschini V, et al. J Org Chem. 2004 Jan 23;69(2):357-73. doi: 10.1021/jo035065+. J Org Chem. 2004. PMID: 14725448

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