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A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4-d]Pyrimidine Dual Src/P-Glycoprotein Inhibitor.
Cancers (Basel). 2019 Jun 19;11(6):848. doi: 10.3390/cancers11060848.
Cancers (Basel). 2019.
PMID: 31248184
Free PMC article.
AuNP Pyrazolo[3,4-d]pyrimidine Nanosystem in Combination with Radiotherapy against Glioblastoma.
Molinari A, Iovenitti G, Mancini A, Gravina GL, Chebbi M, Caruana M, Vignaroli G, Orofino F, Rango E, Angelucci A, Dreassi E, Schenone S, Botta M.
Molinari A, et al. Among authors: rango e.
ACS Med Chem Lett. 2020 Mar 5;11(5):664-670. doi: 10.1021/acsmedchemlett.9b00538. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435368
Free PMC article.
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Si113-prodrugs selectively activated by plasmin against hepatocellular and ovarian carcinoma.
Rango E, D'Antona L, Iovenitti G, Brai A, Mancini A, Zamperini C, Trivisani CI, Marianelli S, Fallacara AL, Molinari A, Cianciusi A, Schenone S, Perrotti N, Dreassi E, Botta M.
Rango E, et al.
Eur J Med Chem. 2021 Nov 5;223:113653. doi: 10.1016/j.ejmech.2021.113653. Epub 2021 Jun 17.
Eur J Med Chem. 2021.
PMID: 34161866
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The Pyrazolo[3,4-d]Pyrimidine Derivative Si306 Encapsulated into Anti-GD2-Immunoliposomes as Therapeutic Treatment of Neuroblastoma.
Rango E, Pastorino F, Brignole C, Mancini A, Poggialini F, Di Maria S, Zamperini C, Iovenitti G, Fallacara AL, Sabetta S, Clementi L, Valoti M, Schenone S, Angelucci A, Ponzoni M, Dreassi E, Botta M.
Rango E, et al.
Biomedicines. 2022 Mar 12;10(3):659. doi: 10.3390/biomedicines10030659.
Biomedicines. 2022.
PMID: 35327462
Free PMC article.
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Focused library of phenyl-fused macrocyclic amidinoureas as antifungal agents.
Balestri LJI, D'Agostino I, Rango E, Vagaggini C, Marchitiello R, Mariotti M, Casian A, Deodato D, Truglio GI, Orofino F, Sanguinetti M, Bugli F, Botta L, Dreassi E.
Balestri LJI, et al. Among authors: rango e.
Mol Divers. 2022 Dec;26(6):3399-3409. doi: 10.1007/s11030-022-10388-7. Epub 2022 Feb 10.
Mol Divers. 2022.
PMID: 35143033
Free PMC article.
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A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery.
Migliorini F, Cini E, Dreassi E, Finetti F, Ievoli G, Macrì G, Petricci E, Rango E, Trabalzini L, Taddei M.
Migliorini F, et al. Among authors: rango e.
Chem Commun (Camb). 2022 Sep 20;58(75):10532-10535. doi: 10.1039/d2cc03052g.
Chem Commun (Camb). 2022.
PMID: 36043993
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Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA.
D'Agostino I, Ardino C, Poli G, Sannio F, Lucidi M, Poggialini F, Visaggio D, Rango E, Filippi S, Petricci E, Visca P, Botta L, Docquier JD, Dreassi E.
D'Agostino I, et al. Among authors: rango e.
Eur J Med Chem. 2022 Mar 5;231:114158. doi: 10.1016/j.ejmech.2022.114158. Epub 2022 Jan 29.
Eur J Med Chem. 2022.
PMID: 35168113
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Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses.
Grazia Martina M, Vicenti I, Bauer L, Crespan E, Rango E, Boccuto A, Olivieri N, Incerti M, Zwaagstra M, Allodi M, Bertoni S, Dreassi E, Zazzi M, van Kuppeveld FJM, Maga G, Radi M.
Grazia Martina M, et al. Among authors: rango e.
ChemMedChem. 2021 Dec 6;16(23):3548-3552. doi: 10.1002/cmdc.202100483. Epub 2021 Sep 7.
ChemMedChem. 2021.
PMID: 34382337
Free PMC article.
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