Rai G - Search Results

1

Inhibition of YAP/TAZ-driven TEAD activity prevents growth of NF2-null schwannoma and meningioma.

Laraba L, Hillson L, de Guibert JG, Hewitt A, Jaques MR, Tang TT, Post L, Ercolano E, Rai G, Yang SM, Jagger DJ, Woznica W, Edwards P, Shivane AG, Hanemann CO, Parkinson DB. Laraba L, et al. Among authors: rai g. Brain. 2023 Apr 19;146(4):1697-1713. doi: 10.1093/brain/awac342. Brain. 2023. PMID: 36148553 Free PMC article.

2

RALDH1 Inhibition Shows Immunotherapeutic Efficacy in Hepatocellular Carcinoma.

Yu P, Cao S, Yang SM, Rai G, Martinez NJ, Yasgar A, Zakharov AV, Simeonov A, Molina Arocho WA, Lobel GP, Mohei H, Scott AL, Zhai L, Furth EE, Simon MC, Haldar M. Yu P, et al. Among authors: rai g. Cancer Immunol Res. 2024 Feb 2;12(2):180-194. doi: 10.1158/2326-6066.CIR-22-1023. Cancer Immunol Res. 2024. PMID: 38051215

3

Real-Time Cellular Thermal Shift Assay to Monitor Target Engagement.

Sanchez TW, Ronzetti MH, Owens AE, Antony M, Voss T, Wallgren E, Talley D, Balakrishnan K, Leyes Porello SE, Rai G, Marugan JJ, Michael SG, Baljinnyam B, Southall N, Simeonov A, Henderson MJ. Sanchez TW, et al. Among authors: rai g. ACS Chem Biol. 2022 Sep 16;17(9):2471-2482. doi: 10.1021/acschembio.2c00334. Epub 2022 Sep 1. ACS Chem Biol. 2022. PMID: 36049119 Free PMC article.

4

Room-Temperature, Copper-Free Sonogashira Reactions Facilitated by Air-Stable, Monoligated Precatalyst [DTBNpP] Pd(crotyl)Cl.

Pohida K, Maloney DJ, Mott BT, Rai G. Pohida K, et al. Among authors: rai g. ACS Omega. 2018 Oct 10;3(10):12985-12998. doi: 10.1021/acsomega.8b01868. eCollection 2018 Oct 31. ACS Omega. 2018. PMID: 31458021 Free PMC article.

5

Target Class Profiling of Small-Molecule Methyltransferases.

Hanson QM, Hoxie N, Shen M, Guo H, Cho IJ, Chakraborty I, Aragon BM, Rai G, Patnaik S, Janiszewski JS, Hall MD. Hanson QM, et al. Among authors: rai g. ACS Chem Biol. 2023 Apr 21;18(4):969-981. doi: 10.1021/acschembio.3c00124. Epub 2023 Mar 28. ACS Chem Biol. 2023. PMID: 36976909 Free PMC article.

6

A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution.

Auld DS, Zhang YQ, Southall NT, Rai G, Landsman M, MacLure J, Langevin D, Thomas CJ, Austin CP, Inglese J. Auld DS, et al. Among authors: rai g. J Med Chem. 2009 Mar 12;52(5):1450-8. doi: 10.1021/jm8014525. J Med Chem. 2009. PMID: 19215089 Free PMC article.

7

Discovery of potent and selective inhibitors of human reticulocyte 15-lipoxygenase-1.

Rai G, Kenyon V, Jadhav A, Schultz L, Armstrong M, Jameson JB, Hoobler E, Leister W, Simeonov A, Holman TR, Maloney DJ. Rai G, et al. J Med Chem. 2010 Oct 28;53(20):7392-404. doi: 10.1021/jm1008852. J Med Chem. 2010. PMID: 20866075 Free PMC article.

8

Discovery of potent and selective inhibitors of human platelet-type 12- lipoxygenase.

Kenyon V, Rai G, Jadhav A, Schultz L, Armstrong M, Jameson JB 2nd, Perry S, Joshi N, Bougie JM, Leister W, Taylor-Fishwick DA, Nadler JL, Holinstat M, Simeonov A, Maloney DJ, Holman TR. Kenyon V, et al. Among authors: rai g. J Med Chem. 2011 Aug 11;54(15):5485-97. doi: 10.1021/jm2005089. Epub 2011 Jul 8. J Med Chem. 2011. PMID: 21739938 Free PMC article.

9

Synthesis, biological evaluation, and structure-activity relationships of a novel class of apurinic/apyrimidinic endonuclease 1 inhibitors.

Rai G, Vyjayanti VN, Dorjsuren D, Simeonov A, Jadhav A, Wilson DM 3rd, Maloney DJ. Rai G, et al. J Med Chem. 2012 Apr 12;55(7):3101-12. doi: 10.1021/jm201537d. Epub 2012 Mar 28. J Med Chem. 2012. PMID: 22455312 Free PMC article.

10

A furoxan-amodiaquine hybrid as a potential therapeutic for three parasitic diseases().

Mott BT, Cheng KC, Guha R, Kommer VP, Williams DL, Vermeire JJ, Cappello M, Maloney DJ, Rai G, Jadhav A, Simeonov A, Inglese J, Posner GH, Thomas CJ. Mott BT, et al. Among authors: rai g. Medchemcomm. 2012 Dec;3(12):1505-1511. doi: 10.1039/C2MD20238G. Medchemcomm. 2012. PMID: 23205265 Free PMC article.

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