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Ligand recognition and allosteric modulation of the human MRGPRX1 receptor.
Nat Chem Biol. 2023 Apr;19(4):416-422. doi: 10.1038/s41589-022-01173-6. Epub 2022 Oct 27.
Nat Chem Biol. 2023.
PMID: 36302898
Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase.
Talibov VO, Fabini E, FitzGerald EA, Tedesco D, Cederfeldt D, Talu MJ, Rachman MM, Mihalic F, Manoni E, Naldi M, Sanese P, Forte G, Lepore Signorile M, Barril X, Simone C, Bartolini M, Dobritzsch D, Del Rio A, Danielson UH.
Talibov VO, et al. Among authors: rachman mm.
Chembiochem. 2021 May 4;22(9):1597-1608. doi: 10.1002/cbic.202000736. Epub 2021 Feb 11.
Chembiochem. 2021.
PMID: 33400854
Free PMC article.
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Predicting how drug molecules bind to their protein targets.
Rachman MM, Barril X, Hubbard RE.
Rachman MM, et al.
Curr Opin Pharmacol. 2018 Oct;42:34-39. doi: 10.1016/j.coph.2018.07.001. Epub 2018 Jul 21.
Curr Opin Pharmacol. 2018.
PMID: 30041063
Review.
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