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A Parallel Synthesis Approach to the Identification of Novel Diheteroarylamide-Based Compounds Blocking HIV Replication: Potential Inhibitors of HIV-1 Pre-mRNA Alternative Splicing.
J Med Chem. 2016 Mar 10;59(5):1869-79. doi: 10.1021/acs.jmedchem.5b01357. Epub 2016 Feb 29.
J Med Chem. 2016.
PMID: 26878150
2-Aminothiazole-4-carboxamides Enhance Readthrough of Premature Termination Codons by Aminoglycosides.
Rabea SM, Baradaran-Heravi A, Balgi AD, Krause A, Hosseini Farahabadi S, Roberge M, Grierson DS.
Rabea SM, et al.
ACS Med Chem Lett. 2019 Apr 9;10(5):726-731. doi: 10.1021/acsmedchemlett.8b00610. eCollection 2019 May 9.
ACS Med Chem Lett. 2019.
PMID: 31097990
Free PMC article.
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A novel class of inhibitors that target SRSF10 and promote p53-mediated cytotoxicity on human colorectal cancer cells.
Sohail M, Shkreta L, Toutant J, Rabea S, Babeu JP, Huard C, Coulombe-Huntington J, Delannoy A, Placet M, Geha S, Gendron FP, Boudreau F, Tyers M, Grierson DS, Chabot B.
Sohail M, et al.
NAR Cancer. 2021 May 25;3(2):zcab019. doi: 10.1093/narcan/zcab019. eCollection 2021 Jun.
NAR Cancer. 2021.
PMID: 34316707
Free PMC article.
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Spirohydantoins and 1,2,4-triazole-3-carboxamide derivatives as inhibitors of histone deacetylase: Design, synthesis, and biological evaluation.
Aboeldahab AMA, Beshr EAM, Shoman ME, Rabea SM, Aly OM.
Aboeldahab AMA, et al. Among authors: rabea sm.
Eur J Med Chem. 2018 Feb 25;146:79-92. doi: 10.1016/j.ejmech.2018.01.021. Epub 2018 Jan 12.
Eur J Med Chem. 2018.
PMID: 29396364
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Synthesis of 5-phenyl-1-(3-pyridyl)-1H-1,2,4-triazole-3-carboxylic acid derivatives of potential anti-inflammatory activity.
Rabea SM, El-Koussi NA, Hassan HY, Aboul-Fadl T.
Rabea SM, et al.
Arch Pharm (Weinheim). 2006 Jan;339(1):32-40. doi: 10.1002/ardp.200500151.
Arch Pharm (Weinheim). 2006.
PMID: 16411174
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Synthesis and antimicrobial evaluation of new nitric oxide-donating fluoroquinolone/oxime hybrids.
Aziz HA, Moustafa GAI, Abuo-Rahma GEA, Rabea SM, Hauk G, Krishna VS, Sriram D, Berger JM, Abbas SH.
Aziz HA, et al. Among authors: rabea sm.
Arch Pharm (Weinheim). 2021 Jan;354(1):e2000180. doi: 10.1002/ardp.202000180. Epub 2020 Sep 21.
Arch Pharm (Weinheim). 2021.
PMID: 32959443
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