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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
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2016 | 1 |
2018 | 3 |
2019 | 1 |
2020 | 1 |
2021 | 1 |
2024 | 0 |
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Page 1
Rapid Optimization of the Metabolic Stability of a Human Immunodeficiency Virus Type-1 Capsid Inhibitor Using a Multistep Computational Workflow.
J Med Chem. 2021 Apr 8;64(7):3747-3766. doi: 10.1021/acs.jmedchem.0c01810. Epub 2021 Mar 22.
J Med Chem. 2021.
PMID: 33750123
Free PMC article.
Composition and Orientation of the Core Region of Novel HIV-1 Entry Inhibitors Influences Metabolic Stability.
Karadsheh R, Meuser ME, Cocklin S.
Karadsheh R, et al.
Molecules. 2020 Mar 21;25(6):1430. doi: 10.3390/molecules25061430.
Molecules. 2020.
PMID: 32245167
Free PMC article.
Item in Clipboard
Field-Based Affinity Optimization of a Novel Azabicyclohexane Scaffold HIV-1 Entry Inhibitor.
Meuser ME, Rashad AA, Ozorowski G, Dick A, Ward AB, Cocklin S.
Meuser ME, et al.
Molecules. 2019 Apr 22;24(8):1581. doi: 10.3390/molecules24081581.
Molecules. 2019.
PMID: 31013646
Free PMC article.
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Exploring Modifications of an HIV-1 Capsid Inhibitor: Design, Synthesis, and Mechanism of Action.
Xu JP, Francis AC, Meuser ME, Mankowski M, Ptak RG, Rashad AA, Melikyan GB, Cocklin S.
Xu JP, et al.
J Drug Des Res. 2018;5(2):1070. Epub 2018 Aug 13.
J Drug Des Res. 2018.
PMID: 30393786
Free PMC article.
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Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library.
Wu G, Zalloum WA, Meuser ME, Jing L, Kang D, Chen CH, Tian Y, Zhang F, Cocklin S, Lee KH, Liu X, Zhan P.
Wu G, et al.
Eur J Med Chem. 2018 Oct 5;158:478-492. doi: 10.1016/j.ejmech.2018.09.029. Epub 2018 Sep 11.
Eur J Med Chem. 2018.
PMID: 30243152
Free PMC article.
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Kinetic Characterization of Novel HIV-1 Entry Inhibitors: Discovery of a Relationship between Off-Rate and Potency.
Meuser ME, Murphy MB, Rashad AA, Cocklin S.
Meuser ME, et al.
Molecules. 2018 Aug 3;23(8):1940. doi: 10.3390/molecules23081940.
Molecules. 2018.
PMID: 30081466
Free PMC article.
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Phosphorylation of the RNA-binding protein Dazl by MAPKAP kinase 2 regulates spermatogenesis.
Williams PA, Krug MS, McMillan EA, Peake JD, Davis TL, Cocklin S, Strochlic TI.
Williams PA, et al.
Mol Biol Cell. 2016 Aug 1;27(15):2341-50. doi: 10.1091/mbc.E15-11-0773. Epub 2016 Jun 8.
Mol Biol Cell. 2016.
PMID: 27280388
Free PMC article.
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