Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Filters
Results by year
Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2017 | 1 |
2018 | 1 |
2019 | 1 |
2020 | 2 |
2022 | 2 |
2024 | 0 |
Search Results
6 results
Results by year
Filters applied: . Clear all
Page 1
Malaria Box-Inspired Discovery of N-Aminoalkyl-β-carboline-3-carboxamides, a Novel Orally Active Class of Antimalarials.
ACS Med Chem Lett. 2022 Feb 23;13(3):365-370. doi: 10.1021/acsmedchemlett.1c00663. eCollection 2022 Mar 10.
ACS Med Chem Lett. 2022.
PMID: 35300096
Free PMC article.
Enantiopure Benzofuran-2-carboxamides of 1-Aryltetrahydro-β-carbolines Are Potent Antimalarials In Vitro.
Almolhim H, Ding S, Butler JH, Bremers EK, Butschek GJ, Slebodnick C, Merino EF, Rizopoulos Z, Totrov M, Cassera MB, Carlier PR.
Almolhim H, et al.
ACS Med Chem Lett. 2022 Feb 24;13(3):371-376. doi: 10.1021/acsmedchemlett.1c00697. eCollection 2022 Mar 10.
ACS Med Chem Lett. 2022.
PMID: 35300082
Free PMC article.
Item in Clipboard
Probing the B- & C-rings of the antimalarial tetrahydro-β-carboline MMV008138 for steric and conformational constraints.
Ding S, Ghavami M, Butler JH, Merino EF, Slebodnick C, Cassera MB, Carlier PR.
Ding S, et al.
Bioorg Med Chem Lett. 2020 Nov 15;30(22):127520. doi: 10.1016/j.bmcl.2020.127520. Epub 2020 Sep 6.
Bioorg Med Chem Lett. 2020.
PMID: 32898696
Free PMC article.
Item in Clipboard
In vitro and in vivo evaluation of the antimalarial MMV665831 and structural analogs.
Ding S, Fike KR, Klemba M, Carlier PR.
Ding S, et al.
Bioorg Med Chem Lett. 2020 Sep 1;30(17):127348. doi: 10.1016/j.bmcl.2020.127348. Epub 2020 Jun 24.
Bioorg Med Chem Lett. 2020.
PMID: 32738996
Free PMC article.
Item in Clipboard
Questioning the γ-gauche effect: stereoassignment of 1,3-disubstituted-tetrahydro-β-carbolines using 1H-1H coupling constants.
Cagašová K, Ghavami M, Yao ZK, Carlier PR.
Cagašová K, et al.
Org Biomol Chem. 2019 Jul 21;17(27):6687-6698. doi: 10.1039/c9ob01139k. Epub 2019 Jun 24.
Org Biomol Chem. 2019.
PMID: 31232413
Free PMC article.
Item in Clipboard
Biological Studies and Target Engagement of the 2- C-Methyl-d-Erythritol 4-Phosphate Cytidylyltransferase (IspD)-Targeting Antimalarial Agent (1 R,3 S)-MMV008138 and Analogs.
Ghavami M, Merino EF, Yao ZK, Elahi R, Simpson ME, Fernández-Murga ML, Butler JH, Casasanta MA, Krai PM, Totrov MM, Slade DJ, Carlier PR, Cassera MB.
Ghavami M, et al.
ACS Infect Dis. 2018 Apr 13;4(4):549-559. doi: 10.1021/acsinfecdis.7b00159. Epub 2017 Nov 7.
ACS Infect Dis. 2018.
PMID: 29072835
Free PMC article.
Item in Clipboard
Cite
Cite