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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2015 | 1 |
2016 | 1 |
2018 | 1 |
2019 | 4 |
2020 | 2 |
2021 | 1 |
2024 | 0 |
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7 results
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Page 1
Medulloblastoma drugs in development: Current leads, trials and drawbacks.
Eur J Med Chem. 2021 Apr 5;215:113268. doi: 10.1016/j.ejmech.2021.113268. Epub 2021 Feb 8.
Eur J Med Chem. 2021.
PMID: 33636537
Free PMC article.
Review.
Inhibition of hedgehog signaling by stereochemically defined des-triazole itraconazole analogues.
Wen J, Teske KA, Kyle Hadden M.
Wen J, et al.
Bioorg Med Chem Lett. 2020 Jan 15;30(2):126794. doi: 10.1016/j.bmcl.2019.126794. Epub 2019 Nov 9.
Bioorg Med Chem Lett. 2020.
PMID: 31761657
Free PMC article.
Item in Clipboard
Formulation and evaluation of itraconazole liposomes for Hedgehog pathway inhibition.
Pace JR, Jog R, Burgess DJ, Hadden MK.
Pace JR, et al.
J Liposome Res. 2020 Sep;30(3):305-311. doi: 10.1080/08982104.2019.1668011. Epub 2019 Oct 2.
J Liposome Res. 2020.
PMID: 31576768
Free PMC article.
Item in Clipboard
Structure-Activity Relationships for Itraconazole-Based Triazolone Analogues as Hedgehog Pathway Inhibitors.
Pace JR, Teske KA, Chau LQ, Dash RC, Zaino AM, Wechsler-Reya RJ, Hadden MK.
Pace JR, et al.
J Med Chem. 2019 Apr 25;62(8):3873-3885. doi: 10.1021/acs.jmedchem.8b01283. Epub 2019 Apr 5.
J Med Chem. 2019.
PMID: 30896941
Free PMC article.
Item in Clipboard
Development of posaconazole-based analogues as hedgehog signaling pathway inhibitors.
Teske KA, Dash RC, Morel SR, Chau LQ, Wechsler-Reya RJ, Hadden MK.
Teske KA, et al.
Eur J Med Chem. 2019 Feb 1;163:320-332. doi: 10.1016/j.ejmech.2018.11.056. Epub 2018 Nov 23.
Eur J Med Chem. 2019.
PMID: 30529635
Free PMC article.
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Repurposing the Clinically Efficacious Antifungal Agent Itraconazole as an Anticancer Chemotherapeutic.
Pace JR, DeBerardinis AM, Sail V, Tacheva-Grigorova SK, Chan KA, Tran R, Raccuia DS, Wechsler-Reya RJ, Hadden MK.
Pace JR, et al.
J Med Chem. 2016 Apr 28;59(8):3635-49. doi: 10.1021/acs.jmedchem.5b01718. Epub 2016 Apr 6.
J Med Chem. 2016.
PMID: 27014922
Free PMC article.
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Synthetic Small Molecule Inhibitors of Hh Signaling As Anti-Cancer Chemotherapeutics.
Maschinot CA, Pace JR, Hadden MK.
Maschinot CA, et al.
Curr Med Chem. 2015;22(35):4033-57. doi: 10.2174/0929867322666150827093904.
Curr Med Chem. 2015.
PMID: 26310919
Free PMC article.
Review.
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